| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRM8 |
(2R,4R)-4-amino-1-methylpyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM8 |
(2R,4R)-4-Amino-1-(2-chloro-benzyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM8 |
(2R,4R)-4-amino-1-ethylpyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM8 |
(2R,4R)-4-Amino-1-(2,2-diphenyl-ethyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM8 |
(S)-3,5-Dihydroxyphenylglycine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM8 |
(2S,4S)-2-amino-4-(4,4-diphenylbutyl)pentanedioic acid |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GSK3A |
Flavone |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| GSK3A |
Roscovitine |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| GSK3A |
Lithium Cation |
NA |
2000000 |
NA |
NA |
NA |
NA |
PubChem |
| GSK3A |
Coumarin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| GSK3A |
Flunixin Meglumine |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| GSK3A |
Semaxanib |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| GSK3A |
1-[(4-methoxyphenyl)methyl]-3-[6-(2H-tetrazol-5-yl)-1,3-benzothiazol-2-yl]urea |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GSK3A |
1-[(4-methoxyphenyl)methyl]-3-[4-(2H-tetrazol-5-yl)pyridin-2-yl]urea |
NA |
370000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GSK3A |
1-[(4-Methoxyphenyl)methyl]-3-(6-nitro-1,3-benzothiazol-2-yl)urea |
NA |
220000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GSK3A |
1-(4-Cyanopyridin-2-yl)-3-[(4-methoxyphenyl)methyl]urea |
NA |
1120000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GSK3A |
N-(2,1,3-Benzothiadiazol-5-yl)acetamide |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| GSK3A |
4-Arylmaleimide deriv. 6a |
NA |
529000 |
NA |
NA |
NA |
NA |
TTD |
| GSK3A |
4-Arylmaleimide deriv. 6b |
NA |
216000 |
NA |
NA |
NA |
NA |
TTD |
| GSK3A |
4-Arylmaleimide deriv. 6c |
NA |
216000 |
NA |
NA |
NA |
NA |
TTD |