| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRM7 |
(2S,4R)-2-amino-4-(2-cyanoethyl)pentanedioic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM7 |
(2S,4R)-2-amino-4-[3-(hydroxyamino)-3-oxopropyl]pentanedioic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM7 |
(2S,4R)-2-amino-4-(2-aminoethyl)pentanedioic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM7 |
(2S,4R)-2-amino-4-(3-aminopropyl)pentanedioic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM7 |
[(3S)-3-amino-3-carboxypropyl]-dihydroxy-(4-hydroxy-3-methoxy-5-nitrobenzoyl)phosphanium |
NA |
NA |
NA |
101000 |
NA |
NA |
BindingDB |
| GRM7 |
(2S)-2-amino-4-[hydroxy-[hydroxy-(5-nitrothiophen-3-yl)methyl]phosphoryl]butanoic acid |
NA |
NA |
NA |
418000 |
NA |
NA |
BindingDB|TTD |
| GRM8 |
(2R,4R)-4-Amino-1-naphthalen-1-ylmethyl-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM8 |
2-Amino-4-(2,2-diphenyl-ethyl)-pentanedioic acid |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM8 |
2-Amino-2,3-methano-4-phosphonobutanoic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM8 |
(2S)-2-amino-4-[[(3-cyanophenyl)-hydroxymethyl]-hydroxyphosphoryl]butanoic acid |
NA |
NA |
NA |
219000 |
NA |
NA |
BindingDB|TTD |
| GRM8 |
(2S)-2-amino-4-[hydroxy-[(4-hydroxy-3-nitrophenyl)methyl]phosphoryl]butanoic acid |
NA |
NA |
NA |
277000 |
NA |
NA |
BindingDB|TTD |
| GRM8 |
1-Benzyl-APDC |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM8 |
4-((S)-1-Carboxy-ethylamino)-benzoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GRM8 |
3-[[[(3S)-3-amino-3-carboxypropyl]-hydroxyphosphoryl]-hydroxymethyl]benzoic acid |
NA |
NA |
NA |
125000 |
NA |
NA |
BindingDB|TTD |
| GRM8 |
4-[[[(3S)-3-amino-3-carboxypropyl]-hydroxyphosphoryl]-hydroxymethyl]benzoic acid |
NA |
NA |
NA |
141000 |
NA |
NA |
BindingDB|TTD |
| GRM8 |
3-[[[(3S)-3-amino-3-carboxypropyl]-hydroxyphosphoryl]methyl]benzoic acid |
NA |
NA |
NA |
511000 |
NA |
NA |
BindingDB|TTD |
| GRM8 |
(2R,4R)-4-Amino-1-(3-chloro-benzyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM8 |
(2R,4R)-4-Amino-1-biphenyl-2-ylmethyl-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM8 |
(2R,4R)-4-Amino-1-naphthalen-2-ylmethyl-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM8 |
(2R,4R)-4-Amino-1-(2,6-dichloro-benzyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |