| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRM6 |
2-Amino-5-(3-hydroxy-5-methyl-isoxazol-4-yl)-pentanoic acid |
NA |
NA |
NA |
410000 |
NA |
NA |
BindingDB|TTD |
| GRM6 |
1-Amino-2,3-dihydro-5-phosphono-1H-indene-1-carboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM6 |
(2R,4R)-4-aminopyrrolidine-2,4-dicarboxylic acid |
110000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRM6 |
Aspartic Acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
PubChem|TTD |
| GRM6 |
(R)-Ampa |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM6 |
2-Aminooctanedioic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM6 |
D-Aspartic Acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
PubChem|TTD |
| GRM6 |
L-2-Aminoadipic Acid |
NA|140000 |
NA |
NA |
140000|NA |
NA |
NA |
BindingDB|PubChem|TTD |
| GRM7 |
2-Amino-4-(2,2-diphenyl-ethyl)-pentanedioic acid |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM7 |
(1S,3R)-1-aminocyclopentane-1,3-dicarboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM7 |
(2S,1''R,2''S)-2-(2''-phosphonocyclopropyl)glycine |
NA |
NA |
NA |
700000 |
NA |
NA |
BindingDB|TTD |
| GRM7 |
(1S,2S)-1-amino-2-(carboxymethyl)cyclopropane-1-carboxylic Acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM7 |
2-Amino-2,3-methano-4-phosphonobutanoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM7 |
(2S)-2-amino-4-[hydroxy-[(R)-hydroxy-(4-hydroxy-3-nitrophenyl)methyl]phosphoryl]butanoic acid |
NA |
NA |
NA |
295000 |
NA |
NA |
BindingDB|TTD |
| GRM7 |
(2S)-2-amino-4-[hydroxy-[hydroxy-(5-nitrofuran-2-yl)methyl]phosphoryl]butanoic acid |
NA |
NA |
NA |
1970000 |
NA |
NA |
BindingDB|TTD |
| GRM7 |
2-amino-2-[(1R,2R,3S)-2-phenyl-3-phosphonocyclopropyl]acetic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM7 |
(1S,2R)-1-amino-2-phosphonomethylcyclopropane-carboxylic acid |
NA |
NA |
NA |
602000 |
NA |
NA |
BindingDB|TTD |
| GRM7 |
(1S,2S)-1-amino-2-phosphonomethylcyclopropane-carboxylic acid |
NA |
NA |
NA |
625000 |
NA |
NA |
BindingDB|TTD |
| GRM7 |
(1R,2S)-1-amino-2-(phosphonomethyl)cyclopropanecarboxylic acid |
NA |
NA |
NA |
3000000 |
NA |
NA |
TTD |
| GRM7 |
(2S)-2-amino-4-phosphonobutanoic acid |
NA|175000 |
NA |
NA |
188000|200000|249000|337000|NA|175000 |
NA |
NA |
BindingDB|GtoPDB|TTD |