| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRM5 |
Amino-(2-chloro-3,5-dihydroxy-phenyl)-acetic acid(S-CHPG) |
10000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
(2S)-2-amino-3-(3,5-dioxo-1,2,4-oxadiazolidin-4-yl)-2-methylpropanoic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRM5 |
2-Amino-bicyclo[3.2.0]heptane-2,7-dicarboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
(2S)-3-(3''-Carboxybicyclo[1.1.1]pentyl)alanine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
(2R)-3-(3''-Carboxybicyclo[1.1.1]pentyl)alanine |
336000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRM5 |
(2S)-2-(3''-Carboxymethylbicyclo[1.1.1]pentyl)glycine |
293000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRM5 |
(2R)-2-(3''-Carboxymethylbicyclo[1.1.1]pentyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
(2S)-(3''-Phosphonomethylbicyclo[1.1.1]pentyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
(2R)-(3'-Phosphonomethylbicyclo[1.1.1]pentyl)glycine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
(RS)-Ppg |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
1-Amino-2,3-dihydro-5-phosphono-1H-indene-1-carboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
(2R,4R)-4-amino-1-benzhydrylpyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
(S)-(+)-Cbpg |
NA|103000 |
NA |
NA |
103000|NA |
NA |
NA |
BindingDB|TTD |
| GRM5 |
4-[(S)-amino(carboxy)methyl]-3-methylbenzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
(S)-4Cpg |
NA |
155000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRM5 |
(2S,4S)-2-amino-4-(4,4-diphenylbutyl)pentanedioic acid |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
(R)-1-Amino-indan-1,5-dicarboxylic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
(1S,3S)-1-aminocyclopentane-1,3-dicarboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM5 |
2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-butyric acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
L-2-Aminoadipic Acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
PubChem|TTD |