| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRM5 |
N-(4-chloro-2-((3,5-dichloro-N-ethylbenzamido)methyl)phenyl)picolinamide |
NA |
NA |
NA |
470000 |
NA |
NA |
BindingDB|TTD |
| GRM5 |
Ctep |
NA |
539000 |
NA |
NA |
NA |
NA |
BindingDB |
| GRM5 |
(1S,2S)-1-amino-2-(carboxymethyl)cyclopropane-1-carboxylic Acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM5 |
Alpha-methyl-4-carboxyphenylglycine, (+/-)- |
2000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
N-(3-fluorophenyl)-3-((2-methylthiazol-4-yl)ethynyl)benzamide |
NA |
133000 |
NA |
NA |
NA |
NA |
BindingDB |
| GRM5 |
N-(3-cyanophenyl)-3-((2-methylthiazol-4-yl)ethynyl)benzamide |
NA |
134000 |
NA |
NA |
NA |
NA |
BindingDB |
| GRM5 |
2-fluoro-N-(4-fluorophenyl)-5-(pyridin-4-ethynyl)benzamide |
NA |
382000 |
NA |
NA |
NA |
NA |
BindingDB |
| GRM5 |
N-(4-fluorophenyl)-2-methyl-5-((2-methyl-thiazol-4-yl)ethynyl)benzamide |
NA |
108500 |
NA |
NA |
NA |
NA |
BindingDB |
| GRM5 |
N-(4-fluorophenyl)-2-methyl-5-(pyridin-2-ethynyl)benzamide |
NA |
104100 |
NA |
NA |
NA |
NA |
BindingDB |
| GRM5 |
3-(2,3-Difluoro-4-methoxyphenyl)-2,5-dimethyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine |
NA |
NA |
NA |
10000000 |
NA |
NA |
TTD |
| GRM5 |
1-Benzyl-APDC |
600000|NA |
NA|300000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRM5 |
(S)-2-amino-5-phosphonopentanoic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
(2R,1''R,2''S)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
(2S,1''S,2''S)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
(2R,1''S,2''S)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
(2S,1''R,2''R)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
(2S)-2-amino-4-phosphonobutanoic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
Aida |
1000000 |
NA |
NA |
NA |
NA |
NA |
PubChem|TTD |
| GRM5 |
3-[Amino(carboxy)methyl]bicyclo[1.1.1]pentane-1-carboxylic acid |
NA |
NA |
NA |
103000 |
NA |
NA |
BindingDB|TTD |
| GRM5 |
4-((S)-1-Carboxy-ethylamino)-benzoic acid |
NA |
195000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |