| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRM4 |
(2R,4R)-4-aminopyrrolidine-2,4-dicarboxylic acid |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
(S)-(+)-Cbpg |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
(2S,3S,4S)-2-Methyl-2-(carboxycyclopropyl)glycine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
(S)-4Cpg |
838000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
(2S)-2-amino-4-[hydroxy-[hydroxy-(4-morpholin-4-yl-3-nitrophenyl)methyl]phosphoryl]butanoic acid |
NA |
NA |
NA |
241000 |
NA |
NA |
TTD |
| GRM4 |
(2S,4S)-2-amino-4-(4,4-diphenylbutyl)pentanedioic acid |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-butyric acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
(1R,2S,3R)-2-[(S)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
280000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
(+/-)-1-Aminocyclopentane-trans-1,3-dicarboxylic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM4 |
L-2-Aminoadipic Acid |
3000000|NA |
NA |
NA |
NA|3000000 |
NA |
NA |
PubChem|TTD |
| GRM4 |
2-Amino-4-(4-hydroxy-[1,2,5]thiadiazol-3-yl)-butyric acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM4 |
Iflwvshrwaivqf-sgihwfkdsa- |
280000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
(S)-Hibo |
490000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRM5 |
4-(amino-carboxy-methyl)-2-hydroxy-5-methyl-benzoic Acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
3-[(R)-amino(carboxy)methyl]bicyclo[1.1.1]pentane-1-carboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM5 |
(2R,4R)-1,4-Diamino-pyrrolidine-2,4-dicarboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
(2R,4R)-4-Amino-1-naphthalen-1-ylmethyl-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
2-Amino-4-(2,2-diphenyl-ethyl)-pentanedioic acid |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM5 |
(1R,2S,4R,5S)-2-Amino-bicyclo[2.1.1]hexane-2,5-dicarboxylic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM5 |
(2S)-2-amino-4-(4-oxo-1,2,5-thiadiazol-3-yl)butanoic acid |
NA |
NA |
NA |
190000 |
NA |
NA |
TTD |