| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRM4 |
(S)-Ampa |
NA |
NA |
NA |
3000000 |
NA |
NA |
TTD |
| GRM4 |
Benzylamino-(3-hydroxy-isoxazol-5-yl)-acetic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM4 |
(S)-2-amino-5-phosphonopentanoic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
alpha-Amino-3-(hydroxy)-5-methyl-4-isoxazoleacetic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM4 |
(2S,1''R,2''S)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
(2R,1''S,2''R)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
(2R,1''R,2''S)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
(2R,1''R,2''R)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
(2S,1''S,2''S)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
(2S,1''S,2''R)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
(2R,1''S,2''S)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
(2S,1''R,2''R)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
Aida |
1000000 |
NA |
NA |
NA |
NA |
NA |
PubChem|TTD |
| GRM4 |
4-((S)-1-Carboxy-ethylamino)-benzoic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
(2S,4S)-4-Methylglutamic acid |
470000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
Quisqualic Acid |
112000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
homo-AMPA |
NA |
NA |
NA |
3000000 |
NA |
NA |
TTD |
| GRM4 |
4-Methylene-L-glutamic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
(2R,4R)-4-Amino-1-(3-chloro-benzyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
(2R,4R)-4-Amino-1-biphenyl-2-ylmethyl-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |