| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRM3 |
(2R,4R)-4-Amino-1-cyclohexylmethyl-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM3 |
(2R,4R)-4-Amino-1-(4-chloro-benzyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM3 |
(1S,2R)-1-amino-2-(carboxymethyl)cyclopropane-1-carboxylic acid |
199526.23 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM3 |
(RS)-Ppg |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM3 |
(2R,4R)-4-amino-1-benzhydrylpyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM3 |
2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-butyric acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM3 |
4,8-Dicarboxy-6-oxo-undecanedioic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM4 |
(S)-Hibo |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
(1S,3R)-1-amino-3-(carboxymethyl)cyclopentane-1-carboxylic Acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
Pccg-13 |
280000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
Ethylamino-(3-hydroxy-isoxazol-5-yl)-acetic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM4 |
(1S,2R,3R)-2-[(S)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
280000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
3-[(R)-amino(carboxy)methyl]bicyclo[1.1.1]pentane-1-carboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM4 |
(S)-2-Amino-3-(4-butyl-3-hydroxy-isoxazol-5-yl)-propionic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
(2R,4R)-1,4-Diamino-pyrrolidine-2,4-dicarboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
(2R,4R)-4-Amino-1-naphthalen-1-ylmethyl-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
2-Amino-4-(2,2-diphenyl-ethyl)-pentanedioic acid |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM4 |
(3-Hydroxy-isoxazol-5-yl)-methylamino-acetic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM4 |
(1R,2S,4R,5S)-2-Amino-bicyclo[2.1.1]hexane-2,5-dicarboxylic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM4 |
(2S)-2-amino-4-(4-oxo-1,2,5-thiadiazol-3-yl)butanoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |