| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRM2 |
(S)-(+)-Cbpg |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(S)-4Cpg |
577000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
Aspartic Acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
PubChem|TTD |
| GRM2 |
(R)-Ampa |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM2 |
2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-butyric acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(1R,2S,3R)-2-[(S)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM2 |
(+/-)-1-Aminocyclopentane-trans-1,3-dicarboxylic acid |
NA |
NA |
NA |
110000 |
NA |
NA |
TTD |
| GRM2 |
2-Aminooctanedioic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM2 |
D-Aspartic Acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
PubChem|TTD |
| GRM2 |
Iflwvshrwaivqf-sgihwfkdsa- |
NA |
NA |
NA |
122000 |
NA |
NA |
TTD |
| GRM3 |
(1S,2S)-1-amino-2-(carboxymethyl)cyclopropane-1-carboxylic Acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM3 |
3-(2,3-Difluoro-4-methoxyphenyl)-2,5-dimethyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine |
NA |
NA |
NA |
10000000 |
NA |
NA |
TTD |
| GRM3 |
1-Benzyl-APDC |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM3 |
(2S)-2-amino-4-phosphonobutanoic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM3 |
(2S,4R)-4-(2,2-Diphenylethylamino-3-oxopropyl)glutamic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GRM3 |
(2R,4R)-4-Amino-1-(3-chloro-benzyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM3 |
(2R,4R)-4-Amino-1-naphthalen-2-ylmethyl-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM3 |
(2R,4R)-4-Amino-1-(2-chloro-benzyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM3 |
(2R,4R)-4-Amino-1-biphenyl-4-ylmethyl-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM3 |
(2R,4R)-4-Amino-1-phenethyl-pyrrolidine-2,4-dicarboxylic acid |
NA |
166000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |