| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRM2 |
(2R,1''S,2''R)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(2R,1''R,2''S)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(2R,1''R,2''R)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(2S,1''S,2''S)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(2S,1''S,2''R)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(2R,1''S,2''S)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(2S,1''R,2''R)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(2S)-2-amino-4-phosphonobutanoic acid |
129000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(3-Amino-3-methyl-butyl)-phosphonic acid(MAP4) |
447000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
Aida |
1000000 |
NA |
NA |
NA |
NA |
NA |
PubChem|TTD |
| GRM2 |
4-((S)-1-Carboxy-ethylamino)-benzoic acid |
NA |
339000 |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(A+-)-1-Amino-cis-cyclopentane-1,3-dicarboxylic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM2 |
D-Glutamic Acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
PubChem|TTD |
| GRM2 |
(2S,4R)-4-(2,2-Diphenylethylamino-3-oxopropyl)glutamic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(2S,3S)-3-(carboxymethyl)azetidine-2-carboxylic acid |
NA |
NA |
NA |
600000 |
NA |
NA |
TTD |
| GRM2 |
Quisqualic Acid |
113000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
homo-AMPA |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM2 |
(2R,4R)-4-Amino-1-(3-chloro-benzyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(2R,4R)-4-amino-1-methylpyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(2R,4R)-4-amino-1-ethylpyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |