| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRM1 |
Iflwvshrwaivqf-sgihwfkdsa- |
135000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(S)-Hibo |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(1S,3R)-1-amino-3-(carboxymethyl)cyclopentane-1-carboxylic Acid |
122000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
Pccg-13 |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM2 |
Ethylamino-(3-hydroxy-isoxazol-5-yl)-acetic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM2 |
2-Aminoheptanedioic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM2 |
(1S,2R,3R)-2-[(S)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM2 |
3-[(R)-amino(carboxy)methyl]bicyclo[1.1.1]pentane-1-carboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM2 |
1-Amino-3-phosphono-3-cyclopentene-1-carboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM2 |
(S)-2-Amino-3-(4-butyl-3-hydroxy-isoxazol-5-yl)-propionic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(3-Hydroxy-isoxazol-5-yl)-methylamino-acetic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM2 |
1-Amino-3-phosphono-2-cyclopentene-1-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(1R,2S,4R,5S)-2-Amino-bicyclo[2.1.1]hexane-2,5-dicarboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM2 |
(1R,2R,3S)-2-[(S)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM2 |
(1S,2R,3S)-2-[(R)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM2 |
(1R,2S,3R)-2-[(R)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM2 |
(1S,2S,3S)-2-[(R)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM2 |
(1S,2S,3S)-2-[(S)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM2 |
2-Amino-6-(3-hydroxy-5-methyl-isoxazol-4-yl)-hexanoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM2 |
(1S,2S)-4-aminocyclopentane-1,2,4-tricarboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |