| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRM2 |
(1R,2R,3R)-2-[(R)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM2 |
(1S,2R,3R)-2-[(R)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM2 |
(1S,2S,3R)-2-[(R)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM2 |
(1S,2R,3S)-2-[(S)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM2 |
(1R,2R,3R)-2-[(S)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM2 |
(1R,4S,5R,6S)-3-azabicyclo[3.3.0]octane-4,6-dicarboxylic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM2 |
(2S,1''R,2''S)-2-(2''-phosphonocyclopropyl)glycine |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM2 |
(1R,2S)-1-amino-2-[(4-oxo-1,2,5-thiadiazol-3-yl)methyl]cyclopropane-1-carboxylic acid;hydrochloride |
NA |
NA |
NA |
251000 |
NA |
NA |
TTD |
| GRM2 |
2-Amino-2-(3-hydroxyphenyl)acetic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
Ibotenic Acid |
110000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
3-(2,3-Difluoro-4-methoxyphenyl)-2,5-dimethyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine |
NA |
NA |
NA |
10000000 |
NA |
NA |
TTD |
| GRM2 |
1-Benzyl-APDC |
NA |
121000 |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(S)-Ampa |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM2 |
Benzylamino-(3-hydroxy-isoxazol-5-yl)-acetic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM2 |
(S)-2-amino-5-phosphonopentanoic acid |
205000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
D-2-aminoadipic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM2 |
2-amino-2-[(1R,2R,3S)-2-phenyl-3-phosphonocyclopropyl]acetic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM2 |
alpha-Amino-3-(hydroxy)-5-methyl-4-isoxazoleacetic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM2 |
L-Homocysteic acid |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(2S,1''R,2''S)-2-(2''-sulfonocyclopropyl)glycine |
235000 |
NA |
NA |
NA |
NA |
NA |
TTD |