| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRM2 |
(2R,4R)-4-Amino-1-(3,3-diphenyl-propyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(2R,4R)-4-Amino-1-(2,4-dichloro-benzyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(2R,4R)-4-Amino-1-biphenyl-4-ylmethyl-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(2R,4R)-4-Amino-1-(3-phenyl-propyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(2R,4R)-4-Amino-1-(4-chloro-benzyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
2-Amino-bicyclo[3.2.0]heptane-2,7-dicarboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
2-Amino-5-(3-hydroxy-5-methyl-isoxazol-4-yl)-pentanoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM2 |
(S)-3,5-Dihydroxyphenylglycine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(S)-2-amino-2-((1R,2S)-2-phosphonocyclopropyl)acetic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM2 |
(S)-2-amino-2-((1S,2R)-2-phosphonocyclopropyl)acetic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM2 |
2-amino-2-[(1S,2S,3R)-2-phenyl-3-phosphonocyclopropyl]acetic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM2 |
2-amino-2-[(1R,2S,3S)-2-phenyl-3-phosphonocyclopropyl]acetic acid |
NA |
NA |
NA |
320000 |
NA |
NA |
TTD |
| GRM2 |
2-amino-2-[(1S,2R,3R)-2-phenyl-3-phosphonocyclopropyl]acetic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM2 |
(2S)-3-(3''-Carboxybicyclo[1.1.1]pentyl)alanine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(2R)-3-(3''-Carboxybicyclo[1.1.1]pentyl)alanine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(2S)-2-(3''-Carboxymethylbicyclo[1.1.1]pentyl)glycine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(2R)-2-(3''-Carboxymethylbicyclo[1.1.1]pentyl)glycine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(RS)-Ppg |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
(2R,4R)-4-amino-1-benzhydrylpyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM2 |
4-Carboxyphenylglycine |
NA |
577000 |
NA |
NA |
NA |
NA |
TTD |