| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRM1 |
(2R)-2-(3''-Carboxymethylbicyclo[1.1.1]pentyl)glycine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2S)-(3''-Phosphonomethylbicyclo[1.1.1]pentyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R)-(3'-Phosphonomethylbicyclo[1.1.1]pentyl)glycine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(RS)-Ppg |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
1-Amino-2,3-dihydro-5-phosphono-1H-indene-1-carboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
Cl-HIBO |
860000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R,4R)-4-amino-1-benzhydrylpyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
Pccg-4 |
270000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
Aspartic Acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
PubChem|TTD |
| GRM1 |
(2S,4S)-2-amino-4-(4,4-diphenylbutyl)pentanedioic acid |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(R)-1-Amino-indan-1,5-dicarboxylic acid |
NA |
214000 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(1S,3S)-1-aminocyclopentane-1,3-dicarboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM1 |
(R)-Ampa |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM1 |
2-Amino-4-(3-hydroxy-5-methyl-isoxazol-4-yl)-butyric acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(1R,2S,3R)-2-[(S)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
270000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(+/-)-1-Aminocyclopentane-trans-1,3-dicarboxylic acid |
NA |
NA |
NA |
127000 |
NA |
NA |
TTD |
| GRM1 |
2-Aminooctanedioic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM1 |
D-Aspartic Acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
PubChem|TTD |
| GRM1 |
L-2-Aminoadipic Acid |
1000000|NA |
NA |
NA |
NA|1000000 |
NA |
NA |
PubChem|TTD |
| GRM1 |
2-Amino-4-(4-hydroxy-[1,2,5]thiadiazol-3-yl)-butyric acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |