| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRM1 |
(2R,4R)-4-Amino-1-naphthalen-2-ylmethyl-pyrrolidine-2,4-dicarboxylic acid |
NA |
133000 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R,4R)-4-Amino-1-(2,6-dichloro-benzyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
238500 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R,4R)-4-Amino-1-(3,4-dichloro-benzyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R,4R)-4-amino-1-methylpyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R,4R)-4-Amino-1-(2-chloro-benzyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R,4R)-4-amino-1-ethylpyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R,4R)-4-Amino-1-(3,3-diphenyl-propyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R,4R)-4-Amino-1-(2,2-diphenyl-ethyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R,4R)-4-Amino-1-(2,4-dichloro-benzyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R,4R)-4-Amino-1-biphenyl-4-ylmethyl-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R,4R)-4-Amino-1-(3-phenyl-propyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R,4R)-4-Amino-1-phenethyl-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R,4R)-4-Amino-1-cyclohexylmethyl-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R,4R)-4-Amino-1-(4-chloro-benzyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
Amino-(2-chloro-3,5-dihydroxy-phenyl)-acetic acid(S-CHPG) |
750000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2S)-2-amino-3-(3,5-dioxo-1,2,4-oxadiazolidin-4-yl)-2-methylpropanoic acid |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
2-Amino-bicyclo[3.2.0]heptane-2,7-dicarboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
2-Amino-5-(3-hydroxy-5-methyl-isoxazol-4-yl)-pentanoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM1 |
(2S)-3-(3''-Carboxybicyclo[1.1.1]pentyl)alanine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R)-3-(3''-Carboxybicyclo[1.1.1]pentyl)alanine |
210000 |
NA |
NA |
NA |
NA |
NA |
TTD |