| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRM1 |
(2S)-2-amino-4-(4-oxo-1,2,5-thiadiazol-3-yl)butanoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM1 |
(1S,2R,3S)-2-[(R)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
270000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(1S,2S,3S)-2-[(R)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
270000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(1S,2S,3S)-2-[(S)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
270000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(1S,2S,4S,5R)-2-Amino-bicyclo[2.1.1]hexane-2,5-dicarboxylic acid |
NA |
NA |
NA |
232000 |
NA |
NA |
TTD |
| GRM1 |
2-Amino-6-(3-hydroxy-5-methyl-isoxazol-4-yl)-hexanoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM1 |
(1S,2S)-4-aminocyclopentane-1,2,4-tricarboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(1R,2R,3R)-2-[(R)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
270000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(1S,2R,3R)-2-[(R)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
270000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(1S,2S,3R)-2-[(R)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
270000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(1S,2R,3S)-2-[(S)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
260000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(1R,2R,3R)-2-[(S)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
205000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(1R,2S,4R,5R)-2-Amino-bicyclo[2.1.1]hexane-2,5-dicarboxylic acid |
NA |
NA |
NA |
121000 |
NA |
NA |
TTD |
| GRM1 |
(1R,4S,5R,6S)-3-azabicyclo[3.3.0]octane-4,6-dicarboxylic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM1 |
(1S,2S)-1-amino-2-(carboxymethyl)cyclopropane-1-carboxylic Acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM1 |
(S)-2-Amino-4-(3,5-dioxo-[1,2,4]oxadiazolidin-2-yl)-butyric acid |
184000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
2-Amino-2-(3-hydroxyphenyl)acetic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
3-(2,3-Difluoro-4-methoxyphenyl)-2,5-dimethyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
1-Benzyl-APDC |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(S)-Ampa |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |