| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRK2 |
N-benzyl-3-[(4-methyl-5-pyridin-4-yl-1,2,4-triazol-3-yl)methylamino]benzamide |
NA |
NA |
NA |
1900000 |
NA |
NA |
BindingDB|TTD |
| GRK2 |
N-[(2-chlorophenyl)methyl]-3-[(3-pyridin-4-yl-1H-1,2,4-triazol-5-yl)methylamino]benzamide |
NA |
NA |
NA |
120000 |
NA |
NA |
BindingDB|TTD |
| GRK2 |
3-[(4-methyl-5-pyridin-4-yl-1,2,4-triazol-3-yl)methylamino]-N-[[3-(trifluoromethyl)phenyl]methyl]benzamide |
NA |
NA |
NA |
220000 |
NA |
NA |
BindingDB|TTD |
| GRK2 |
2-[5-Amino-3-(3,4-dihydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl)-3H-imidazol-4-yl]-acetamide |
NA |
557000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRK2 |
3-(Tert-butyl)-2-propanoylindeno[3,2-C]pyrazol-4-one |
NA |
563000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRK2 |
GRK2 Inhibitor |
NA |
126000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRK2 |
Isoproterenone |
NA |
NA |
900000 |
NA |
NA |
NA |
BindingDB |
| GRK2 |
Defluoro Paroxetine, Hydrochloride |
NA |
316200 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(S)-Hibo |
250000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(1S,3R)-1-amino-3-(carboxymethyl)cyclopentane-1-carboxylic Acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
Pccg-13 |
270000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
2-Aminoheptanedioic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM1 |
(1S,2R,3R)-2-[(S)-amino(carboxy)methyl]-3-phenylcyclopropane-1-carboxylic acid |
270000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
3-[(R)-amino(carboxy)methyl]bicyclo[1.1.1]pentane-1-carboxylic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
TTD |
| GRM1 |
(S)-2-Amino-3-(4-butyl-3-hydroxy-isoxazol-5-yl)-propionic acid |
110000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R,4R)-1,4-Diamino-pyrrolidine-2,4-dicarboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R,4R)-4-Amino-1-naphthalen-1-ylmethyl-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
2-Amino-4-(2,2-diphenyl-ethyl)-pentanedioic acid |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2S,3S,4S)-2-amino-3,4-dihydroxy-pentanedioic Acid |
NA |
NA |
NA |
257000 |
NA |
NA |
TTD |
| GRM1 |
(1R,2S,4R,5S)-2-Amino-bicyclo[2.1.1]hexane-2,5-dicarboxylic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |