Navigator

      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
GRIN1 N-[4-[2-(4-benzylpiperidin-1-yl)propanoyl]phenyl]-2-chloroacetamide NA 230000 NA NA NA NA BindingDB
GRIN1 3-Phenyl-3-piperidin-1-ylpiperidin-2-one NA 158489 NA NA NA NA BindingDB
GRIN1 1-Methyl-3-phenyl-3-piperidin-1-ylpyrrolidin-2-one NA 251189 NA NA NA NA BindingDB
GRIN1 6-bromo-2-oxo-2H-chromene-3-carboxylic acid NA 426000 NA NA NA NA BindingDB
GRIN2A (E)-4-(6-Methoxy-2-(3-nitrostyryl)-4-oxoquinazolin-3(4H)-yl)benzoic acid NA 182000 NA NA NA NA TTD
GRIN2B Spermine NA NA NA 125000|127000 NA NA BindingDB|PubChem|TTD
GRIN2B (2-(methylthio)-4,5-dihydro-1H-imidazol-1-yl)(p-tolyl)methanone NA 174000 NA NA NA NA BindingDB
GRIN2B 4-[(3Z)-5-(4-bromophenyl)-3-(6-methyl-2-oxo-4-phenylquinolin-3-ylidene)pyrazolidin-1-yl]-4-oxobutanoic acid NA 113000 NA NA NA NA TTD
GRIN2B NA 113000 NA NA NA NA BindingDB
GRIN2B (E)-4-(6-Methoxy-2-(3-nitrostyryl)-4-oxoquinazolin-3(4H)-yl)benzoic acid NA 193000 NA NA NA NA BindingDB|TTD
GRIN2B (4-Tert-butylphenyl)-(2-methylsulfanyl-4,5-dihydroimidazol-1-yl)methanone NA 138000 NA NA NA NA BindingDB
GRIN2B 2-Methyl-4-(pyridin-3-ylethynyl)thiazole NA 300000 NA NA NA NA TTD
GRIN2C Pregnenolone sulfate NA 112000 NA NA NA NA BindingDB
GRIN2C (4-Tert-butylphenyl)-(2-methylsulfanyl-4,5-dihydroimidazol-1-yl)methanone NA 139000 NA NA NA NA BindingDB
GRIN2C 2-[(4-Tert-butylbenzoyl)amino]-5-methyl-3-thiophenecarboxylic acid NA 175000 NA NA NA NA BindingDB
GRIN2D Pregnenolone sulfate NA 118000 NA NA NA NA BindingDB
GRIN2D (4-Tert-butylphenyl)-(2-methylsulfanyl-4,5-dihydroimidazol-1-yl)methanone NA 210000 NA NA NA NA BindingDB
GRIN2D 6-bromo-2-oxo-2H-chromene-3-carboxylic acid NA 426000 NA NA NA NA BindingDB|TTD
GRIN2D 2-[(4-Tert-butylbenzoyl)amino]-5-methyl-3-thiophenecarboxylic acid NA 120000 NA NA NA NA BindingDB
GRK2 3-[(4-methyl-5-pyridin-4-yl-1,2,4-triazol-3-yl)methylamino]-N-[[4-(trifluoromethyl)phenyl]methyl]benzamide NA NA NA 930000 NA NA BindingDB|TTD