| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRIA3 |
2-Amino-3-(4-bromo-3-hydroxyisoxazol-5-YL)propanoic acid |
NA |
NA |
NA |
202000 |
NA |
NA |
BindingDB |
| GRIA3 |
Glutamic Acid |
NA |
NA |
NA |
15848900000000 |
NA |
NA |
PubChem |
| GRIA3 |
Cl-HIBO |
NA |
NA |
NA |
2700000 |
NA |
NA |
BindingDB |
| GRIA3 |
6-(4-Carboxy-imidazol-1-ylmethyl)-decahydro-isoquinoline-3-carboxylic acid; hydrochloride |
247000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA4 |
2-Amino-3-[3-hydroxy-5-(1-methyl-1H-tetrazol-5-yl)-isoxazol-4-yl]-propionic acid |
NA |
NA |
NA |
3000000 |
NA |
NA |
BindingDB|TTD |
| GRIA4 |
2-amino-3-(3-hydroxy-5-(2-isopropyl-2H-tetrazol-5-yl)isoxazol-4-yl)propanoic acid |
NA |
NA |
NA |
160000 |
NA |
NA |
BindingDB |
| GRIA4 |
Cx516 |
NA |
NA |
NA |
156000|1000000 |
NA |
NA |
BindingDB|PubChem|TTD |
| GRIA4 |
2-amino-3-(2-ethyl-5-oxo-1H-triazol-4-yl)propanoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRIA4 |
(RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid |
NA |
NA |
NA |
490000 |
NA |
NA |
BindingDB |
| GRIA4 |
Aniracetam |
NA |
NA |
NA |
1000000 |
NA |
NA |
PubChem |
| GRIA4 |
Glutamic Acid |
NA |
NA |
NA |
39810700000000 |
NA |
NA |
PubChem |
| GRIA4 |
6-(4-Carboxy-imidazol-1-ylmethyl)-decahydro-isoquinoline-3-carboxylic acid; hydrochloride |
262000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIK1 |
Tezampanel |
NA |
247000 |
NA |
NA |
NA |
NA |
PubChem |
| GRIK1 |
(3S,4aS,6S,8aR)-6-[2-fluoro-6-(2H-tetrazol-5-yl)phenoxy]-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;hydrochloride |
422000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRIK1 |
(3S,4aR,6S,8aR)-6-(4-carboxyanilino)-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid |
528000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRIK1 |
(3S,4aS,6S,8aR)-6-(4-carboxyphenoxy)-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;hydrochloride |
267000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRIK1 |
(3S,4aS,6S,8aR)-6-(2-carboxy-6-chlorophenoxy)-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;hydrochloride |
316000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRIK1 |
(3S,4aS,6S,8aR)-6-(2-carboxy-6-methylphenoxy)-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;hydrochloride |
228000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRIK2 |
Tezampanel |
NA |
247000 |
NA |
NA |
NA |
NA |
PubChem |
| GRIK2 |
(S)-2-Amino-4-(1-ethyl-propylidene)-pentanedioic acid |
207000 |
NA |
NA |
NA |
NA |
NA |
TTD |