| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRIA2 |
2-amino-3-(3-hydroxy-5-(2-isopropyl-2H-tetrazol-5-yl)isoxazol-4-yl)propanoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
BindingDB |
| GRIA2 |
2-amino-3-(2-methyl-5-oxo-1H-triazol-4-yl)propanoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRIA2 |
4,6-Dimethyl-2,3-dihydro-1lambda6,2,4-benzothiadiazine 1,1-dioxide |
NA |
NA |
NA |
403300|407380 |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
2-amino-3-(2-ethyl-5-oxo-1H-triazol-4-yl)propanoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRIA2 |
(RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid |
NA |
NA |
NA |
3000000 |
NA |
NA |
TTD |
| GRIA2 |
2H-1,2,4-Benzothiadiazine, 3,4-dihydro-4-methyl-, 1,1-dioxide |
NA |
NA |
NA |
176300|177828 |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
Glutamic Acid |
NA |
NA |
NA |
140000|7943280000000 |
NA |
NA |
BindingDB|PubChem |
| GRIA2 |
6-(4-Amino-3,5-dimethylphenyl)-2,3,8,10-tetrahydro-[1,4]dioxino[2,3-h][2,3]benzodiazepin-9-one |
164000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| GRIA2 |
(+)-2-Amino-4-(4-hydroxy-1,2,5-oxadiazol-3-yl)butanoicAcid |
NA |
NA |
NA |
489000 |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
(+)-2-Amino-5-(4-hydroxy-1,2,5-oxadiazol-3-yl)pentanoicAcid |
NA |
NA |
NA |
491000|489778.82 |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
(R)-N-(2-phenylpropyl)methanesulfonamide |
NA |
NA |
NA |
1980000 |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
(3S,4aR,6S,8aR)-6-[3-methyl-2-(2H-tetrazol-5-yl)anilino]-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid |
128000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
(3S,4aR,6S,8aR)-6-[(3-Carboxyphenyl)amino]decahydro-3-isoquinolinecarboxylic acid |
238000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
2-((3-((2S)-2-amino-2-carboxyethyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidin-1-yl)methyl)benzoic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRIA2 |
(3S,4aR,6S,8aR)-6-[(4-carboxyphenyl)methyl]-decahydroisoquinoline-3-carboxylic acid |
553000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| GRIA2 |
(3S,4aS,6S,8aR)-6-(2-carboxy-5-chlorophenoxy)-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;hydrochloride |
151000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
(3S,4aR,6S,8aR)-6-[(4-carboxyphenyl)methyl]-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;hydrochloride |
553000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRIA2 |
(1S,2S,6R,8S)-6-(carboxymethyl)-3-oxo-7-oxa-4,12-diazatricyclo[6.4.0.02,6]dodec-9-ene-5-carboxylic acid |
560000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
(3S,4aS,6S,8aR)-6-[3-methoxy-2-(2H-tetrazol-5-yl)phenoxy]-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;hydrochloride |
252000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
(3S,4aR,6S,8aR)-6-[3-methoxy-2-(2H-tetrazol-5-yl)anilino]-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;hydrochloride |
181000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |