| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRIA2 |
(3S,4aS,6S,8aR)-6-[2-fluoro-6-(2H-tetrazol-5-yl)phenoxy]-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;hydrochloride |
450000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
(3S,4aS,6S,8aR)-6-[5-phenoxy-2-(2H-tetrazol-5-yl)phenoxy]-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;hydrochloride |
335000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
(3S,4aR,6S,8aR)-6-(4-carboxyanilino)-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid |
1420000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
(3S,4aS,6S,8aR)-6-(4-carboxyphenyl)sulfanyl-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid |
418000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
(3S,4aS,6S,8aR)-6-(4-carboxyphenoxy)-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;hydrochloride |
913000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
(3S,4aS,6S,8aR)-6-(2-carboxy-4-methylphenoxy)-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;hydrochloride |
107000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
(3S,4aS,6S,8aR)-6-(2-carboxy-4-phenylphenoxy)-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;hydrochloride |
172000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
(3S,4aS,6S,8aR)-6-(2-carboxy-5-methoxyphenoxy)-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;hydrochloride |
111000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
(3S,4aS,6S,8aR)-6-(2-carboxy-6-chlorophenoxy)-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;hydrochloride |
1470000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
(3S,4aS,6S,8aR)-6-(2-carboxy-6-methylphenoxy)-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;hydrochloride |
818000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
(3S,4aR,6S,8aR)-6-[(2-carboxyphenyl)methyl]-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;hydrochloride |
29600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
(3S,4aR,6S,8aR)-6-[(3-carboxyphenyl)methyl]-1,2,3,4,4a,5,6,7,8,8a-decahydroisoquinoline-3-carboxylic acid;hydrochloride |
149000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
6-(4-Carboxy-imidazol-1-ylmethyl)-decahydro-isoquinoline-3-carboxylic acid; hydrochloride |
117000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA3 |
2-Amino-3-[3-hydroxy-5-(1-methyl-1H-tetrazol-5-yl)-isoxazol-4-yl]-propionic acid |
NA |
NA |
NA |
3000000 |
NA |
NA |
TTD |
| GRIA3 |
(RS)-2-amino-3-[3-hydroxy-5-(2-propyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid |
NA |
NA |
NA |
450000 |
NA |
NA |
BindingDB |
| GRIA3 |
2-amino-3-(3-hydroxy-5-(2-isopropyl-2H-tetrazol-5-yl)isoxazol-4-yl)propanoic acid |
NA |
NA |
NA |
700000 |
NA |
NA |
BindingDB |
| GRIA3 |
2-amino-3-(2-methyl-5-oxo-1H-triazol-4-yl)propanoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRIA3 |
2-amino-3-(2-ethyl-5-oxo-1H-triazol-4-yl)propanoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRIA3 |
(RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
BindingDB|TTD |
| GRIA3 |
Aniracetam |
NA |
NA |
NA |
1000000 |
NA |
NA |
PubChem |