| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRB2 |
4-[(2S)-2-{[(1S)-1-{3-[(3,4-dichlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-3-phenylpropyl]carbamoyl}-2-acetamidoethyl]phenoxyphosphonic acid |
NA |
340000 |
NA |
NA |
NA |
NA |
BindingDB |
| GRB2 |
4-[(2S)-2-{[(1S)-1-{3-[(3,4-dichlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}-2-hydroxyethyl]carbamoyl}-2-(1-phenylacetamido)ethyl]phenoxyphosphonic acid |
NA |
263000 |
NA |
NA |
NA |
NA |
BindingDB |
| GRB2 |
4-[(2S)-2-{[(1S)-2-hydroxy-1-[3-(naphthalen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]ethyl]carbamoyl}-2-(1-phenylacetamido)ethyl]phenoxyphosphonic acid |
NA |
368000 |
NA |
NA |
NA |
NA |
BindingDB |
| GRB2 |
CID 5474940 |
NA |
320000 |
NA |
NA |
NA |
NA |
BindingDB |
| GRB2 |
Sodium 2-(4-(2-(4-phosphonatooxyphenoxy)phenyl)-6-(4-phosphonatooxyphenylamino)-1,3,5-triazin-2-ylamino)acetamide |
NA |
265000 |
NA |
NA |
NA |
NA |
BindingDB |
| GRB7 |
Ac(1)-Ala(indol-2-yl)(indol-2-yl)-Phe-Glu-Gly-Tyr-Asp-Asn-Thr-Phe-Pro-Cys(1)-NH2 |
NA |
NA |
347000 |
NA |
NA |
NA |
BindingDB |
| GRIA1 |
2-Amino-3-[3-hydroxy-5-(1-methyl-1H-tetrazol-5-yl)-isoxazol-4-yl]-propionic acid |
NA |
NA |
NA |
3000000 |
NA |
NA |
TTD |
| GRIA1 |
(RS)-2-amino-3-[3-hydroxy-5-(2-propyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid |
NA |
NA |
NA |
480000 |
NA |
NA |
BindingDB |
| GRIA1 |
2-amino-3-(3-hydroxy-5-(2-isopropyl-2H-tetrazol-5-yl)isoxazol-4-yl)propanoic acid |
NA |
NA |
NA |
550000 |
NA |
NA |
BindingDB |
| GRIA1 |
(2S,4Z)-2-amino-4-(2-methylpropylidene)pentanedioic Acid |
113400 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA1 |
N-[3-[[4-[(3-Aminopropyl)amino]butyl]amino]propyl]-4-hydroxy-alpha-[(1-oxobutyl)amino]benzenepropanamide |
170000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| GRIA1 |
2-amino-3-(2-ethyl-5-oxo-1H-triazol-4-yl)propanoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRIA1 |
2-amino-3-(5-oxo-2-propyl-1H-triazol-4-yl)propanoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRIA1 |
(RS)-2-amino-3-[3-hydroxy-5-(2-benzyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid |
NA |
NA |
NA |
3000000|500000 |
NA |
NA |
BindingDB|TTD |
| GRIA1 |
Glutamic Acid |
NA |
NA |
NA |
15848900000000|125893|140000|110000 |
NA |
NA |
PubChem |
| GRIA1 |
6-(4-Carboxy-imidazol-1-ylmethyl)-decahydro-isoquinoline-3-carboxylic acid; hydrochloride |
134000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
(S)-2-Amino-4-(1-ethyl-propylidene)-pentanedioic acid |
280900 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRIA2 |
4-Ethyl-3,4-dihydro-2H-pyrido[4,3-e][1,2,4]thiadiazine 1,1-dioxide |
NA |
NA |
1200000 |
NA |
NA |
NA |
BindingDB |
| GRIA2 |
2-Amino-3-[3-hydroxy-5-(1-methyl-1H-tetrazol-5-yl)-isoxazol-4-yl]-propionic acid |
NA |
NA |
NA |
3000000 |
NA |
NA |
TTD |
| GRIA2 |
(RS)-2-amino-3-[3-hydroxy-5-(2-propyl-2H-5-tetrazolyl)-4-isoxazolyl]propionic acid |
NA |
NA |
NA |
830000 |
NA |
NA |
BindingDB |