| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GPR35 |
6-Hydroxythieno[3,2-b]thiophene-5-carboxylic acid |
NA |
NA |
NA |
340000 |
NA |
NA |
BindingDB |
| GPR35 |
3-(3,5-difluorophenyl)-5,6-dihydroxy-1H-indole-2-carboxylic acid |
NA |
NA |
NA |
109000 |
NA |
NA |
BindingDB |
| GPR35 |
3-Bromo-6-cyclopropylthieno[3,2-b]thiophene-5-carboxylic acid |
NA |
NA |
NA |
504000 |
NA |
NA |
BindingDB |
| GPR35 |
3-(4-chlorophenyl)-5,6-dihydroxy-1H-indole-2-carboxylic acid |
NA |
NA |
NA |
387000 |
NA |
NA |
BindingDB |
| GPR35 |
3-bromo-6-methyl-4H-thieno[3,2-b]pyrrole-5-carboxylic acid |
NA |
NA |
NA |
113000 |
NA |
NA |
BindingDB |
| GPR37L1 |
3-[(1R,2S,4aS,6S,8aR)-3,4a,6-trimethyl-2-[(2E,4E)-4-methylhexa-2,4-dien-2-yl]-2,5,6,7,8,8a-hexahydro-1H-naphthalene-1-carbonyl]-5-benzyl-5-hydroxy-1H-pyrrol-2-one |
NA |
2500000 |
NA |
NA |
NA |
NA |
BindingDB |
| GPR55 |
Psb-SB-489 |
NA |
NA |
283791903 |
NA |
NA |
NA |
BindingDB |
| GPR55 |
Psb-SB-487 |
NA |
NA |
328851631 |
NA |
NA |
NA |
BindingDB |
| GPR84 |
Setogepram |
NA |
398107 |
NA |
NA |
NA |
NA |
GtoPDB |
| GPR84 |
3-Hydroxydecanoic acid |
NA |
NA |
NA |
230000 |
NA |
NA |
GtoPDB |
| GPR84 |
Setogepram sodium |
NA |
398000|208000 |
NA |
NA |
NA |
NA |
PubChem |
| GPR88 |
(1R,2R)-N-[(1R)-2-hydroxy-1-naphthalen-2-ylethyl]-2-phenylcyclopropane-1-carboxamide |
NA |
NA |
NA |
270000 |
NA |
NA |
TTD |
| GPR88 |
(1S,2R)-N-[(1R)-2-hydroxy-1-naphthalen-2-ylethyl]-2-phenylcyclopropane-1-carboxamide |
NA |
NA |
NA |
110000 |
NA |
NA |
TTD |
| GRB2 |
2-{4-[(S)-2-((S)-2-Acetylamino-3-carbamoyl-propionylamino)-2-((S)-1-{(S)-2-carbamoyl-1-[(1S,2S)-1-((S)-1-carbamoyl-3-carboxy-propylcarbamoyl)-2-methyl-butylcarbamoyl]-ethylcarbamoyl}-2-methyl-propylcarbamoyl)-ethyl]-phenoxy}-malonic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| GRB2 |
Ac(1)-Ala(indol-2-yl)(indol-2-yl)-Phe-Glu-Gly-Tyr-Asp-Asn-Thr-Phe-Pro-Cys(1)-NH2 |
NA |
NA |
200000 |
NA |
NA |
NA |
BindingDB |
| GRB2 |
Ac(1)-Ala(indol-2-yl)(indol-2-yl)-Phe-Glu-Gly-Phe(4-EtO2H)-Asp-Asn-Thr-Phe-Pro-Cys(1)-NH2 |
NA |
NA |
440000 |
NA |
NA |
NA |
BindingDB |
| GRB2 |
Ac(1)-Ala(indol-2-yl)(indol-2-yl)-Phe-Glu-Gly-Phe(4-CO2H)-Asp-Asn-Thr-Phe-Pro-Cys(1)-NH2 |
NA |
NA |
560000 |
NA |
NA |
NA |
BindingDB |
| GRB2 |
N-Fmoc-(3''-CH2CH2CO2H-Tyr)-(alpha-Me)Glu-Asn-amide |
NA |
168000 |
NA |
NA |
NA |
NA |
BindingDB |
| GRB2 |
N-Fmoc-(R)-(alpha-Me)Adi-Leu-(3''-NH2-Tyr)-Ac6c-Asn-amide |
NA |
700000 |
NA |
NA |
NA |
NA |
BindingDB |
| GRB2 |
N-Fmoc-(S)-(alpha-Me)Adi-Leu-Tyr-Ac6c-Asn-amide |
NA |
117700 |
NA |
NA |
NA |
NA |
BindingDB |