| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GP6 |
Honokiol |
NA |
NA |
289000 |
NA |
NA |
NA |
PubChem |
| GPBAR1 |
Dinorursodeoxycholic acid |
NA |
NA |
NA |
316000 |
NA |
NA |
TTD |
| GPBAR1 |
Dehydroepiandrosterone Sulfate |
NA |
NA |
NA |
127000 |
NA |
NA |
BindingDB|PubChem|TTD |
| GPBAR1 |
Avicholic Acid Sodium Salt |
NA |
NA |
NA |
160000 |
NA |
NA |
TTD |
| GPBAR1 |
(E)-4-[2,5-dichloro-4-[3-(4-cyclopropyl-2,3-dihydroquinoxaline-1-carbonyl)pyridin-4-yl]oxyphenyl]but-3-enoic acid |
NA |
NA |
NA |
378000 |
NA |
NA |
BindingDB|TTD |
| GPBAR1 |
(3beta,5beta,9beta)-3-(Acetyloxy)cholan-24-Oic Acid |
NA |
NA |
NA |
102000 |
NA |
NA |
TTD |
| GPBAR1 |
Avicholic acid anion |
NA |
NA |
NA |
160000 |
NA |
NA |
BindingDB |
| GPBAR1 |
Tauroursodeoxycholic acid |
NA |
NA |
NA |
105150 |
NA |
NA |
BindingDB|PubChem |
| GPR119 |
Tert-butyl 4-[5-[(3-methylsulfonylpyridin-4-yl)methoxy]pyrimidin-2-yl]piperazine-1-carboxylate |
NA |
NA |
NA |
30000000 |
NA |
NA |
TTD |
| GPR119 |
3-Fluoro-4-(5-fluoro-6-(4-(3-(2-fluoropropan-2-yl)-1,2,4-oxadiazol-5-yl)piperidin-1-yl)pyrimidin-4-ylamino)benzoic acid |
NA |
NA |
NA |
100000000 |
NA |
NA |
TTD |
| GPR139 |
Phenylalanine |
NA|872000 |
NA |
NA |
320000|NA |
NA |
NA |
GtoPDB |
| GPR139 |
Tryptophan |
NA|738000 |
NA |
NA |
220000|NA |
NA |
NA |
GtoPDB |
| GPR35 |
3,4-Dinitrophenol |
NA |
NA |
NA |
112000 |
NA |
NA |
TTD |
| GPR35 |
2,4-Dinitrophenol |
NA |
NA |
NA |
272000 |
NA |
NA |
PubChem |
| GPR35 |
5,6-Dihydroxy-1-benzothiophene-2-carboxylic acid |
NA |
NA |
NA |
520000 |
NA |
NA |
BindingDB |
| GPR35 |
Kynurenic Acid |
NA|137000 |
NA |
NA |
152000|217000|NA|500000 |
NA |
NA |
BindingDB|PubChem |
| GPR35 |
5,6-Dihydroxy-3-methyl-1-benzofuran-2-carboxylic acid |
NA |
NA |
NA |
133000 |
NA |
NA |
BindingDB |
| GPR35 |
|
NA |
NA |
NA |
277000 |
NA |
NA |
BindingDB |
| GPR35 |
3-cyclopropyl-6-methyl-4H-thieno[3,2-b]pyrrole-5-carboxylic acid |
NA |
NA |
NA |
119000 |
NA |
NA |
BindingDB |
| GPR35 |
3-bromo-5,6-dihydroxy-1H-indole-2-carboxylic acid |
NA |
NA |
NA |
166000 |
NA |
NA |
BindingDB |