Navigator

      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
GLO1 Methyl 3-(2-hydroxy-2-phenylacetyl)sulfanylpropanoate 38600000 NA NA NA NA NA TTD
GLO1 S-butyl 2-hydroxy-2-phenylethanethioate 29600000 NA NA NA NA NA TTD
GLO1 Fenoprofen 383000|400000 NA NA NA NA NA PubChem|TTD
GLO1 N-(quinolin-8-yl)acetamide NA 200000 NA NA NA NA TTD
GLO1 Ketoprofen 843000|843100|414000 NA NA NA NA NA PubChem|TTD
GLO1 2-Amino-5-[[1-[(2-ethoxy-2-oxoethyl)amino]-5-[hydroxy(methyl)amino]-1,5-dioxopentan-2-yl]amino]-5-oxopentanoic acid NA 140500 NA NA NA NA TTD
GLO1 2-Amino-5-[[1-[(2-ethoxy-2-oxoethyl)amino]-5-(hydroxyamino)-1,5-dioxopentan-2-yl]amino]-5-oxopentanoic acid NA 1624600 NA NA NA NA TTD
GLO1 2-[(3-Nitrophenyl)methylidene]propanedioic acid 426000 NA NA NA NA NA TTD
GLO1 (2S)-2-amino-5-[[1-(carboxymethylamino)-1-oxo-3-phenacylsulfanylpropan-2-yl]amino]-5-oxopentanoic acid 194984.46 NA NA NA NA NA TTD
GLO1 (2S)-2-amino-5-[[1-(carboxymethylamino)-3-[2-(4-hydroxyphenyl)-2-oxoethyl]sulfanyl-1-oxopropan-2-yl]amino]-5-oxopentanoic acid 194984.46 NA NA NA NA NA TTD
GLO1 (2S)-2-amino-5-[[3-[2-(4-aminophenyl)-2-oxoethyl]sulfanyl-1-(carboxymethylamino)-1-oxopropan-2-yl]amino]-5-oxopentanoic acid 436515.83 NA NA NA NA NA TTD
GLO1 glutaryl-DL-Cys(Bn(4-Br))(Bn(4-Br))-Gly-OH 269153.48 NA NA NA NA NA TTD
GLO1 2-Amino-3-(propanoylsulfanylmethyl)butanedioic acid 1980000 NA NA NA NA NA TTD
GLO1 S-(N-Methyl-N-hydroxycarbomyl)glutathione 680000 NA NA NA NA NA TTD
GLO1 2-azaniumyl-4-ethoxy-3-[[(2R)-2-hydroxypropanoyl]sulfanylmethyl]-4-oxobutanoate 3160000 NA NA NA NA NA TTD
GLO1 2-amino-3-[[(2R)-2-hydroxypropanoyl]sulfanylmethyl]butanedioic acid 2230000 NA NA NA NA NA TTD
GLO1 2-Amino-3-(methylcarbamoylsulfanylmethyl)butanedioic acid 5670000 NA NA NA NA NA TTD
GLO1 N-quinolin-5-ylmethanesulfonamide NA 200000 NA NA NA NA TTD
GLO1 8-Quinolinyl mesylate NA 200000 NA NA NA NA TTD
GLO1 Ethyl 2-(4-nitrobenzylidene)-3-oxobutanoate 159000 NA NA NA NA NA TTD