| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GLB1 |
1-beta-d-Galactosyl-4-phenyl triazole |
330000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GLB1 |
(1S,2S,3S,6R)-6-(3-hydroxypropylamino)cyclohex-4-ene-1,2,3-triol;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GLB1 |
(1S,2S,3S,6R)-6-(cyclohexylamino)cyclohex-4-ene-1,2,3-triol;hydrochloride |
NA |
490000 |
NA |
NA |
NA |
NA |
TTD |
| GLB1 |
(1S,2S,3S,6R)-6-(pentan-3-ylamino)cyclohex-4-ene-1,2,3-triol;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GLB1 |
(1S,2S,3S,6R)-6-(benzylamino)cyclohex-4-ene-1,2,3-triol;hydrochloride |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| GLB1 |
(1S,2S,3S,6R)-6-(octylamino)cyclohex-4-ene-1,2,3-triol;hydrochloride |
NA |
120000 |
NA |
NA |
NA |
NA |
TTD |
| GLB1 |
(3R,4S)-pyrrolidine-3,4-diol |
NA |
720000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GLB1 |
N,N'-Bis(salicylideneamino)oxamide |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| GLB1 |
(3R,4S,5S,6S)-5-(hydroxymethyl)-6-pentylpiperidine-3,4-diol |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| GLB1 |
3-Hydroxy-4-((2-hydroxynaphthyl)azo)naphthalene-1-sulphonic acid |
NA |
600000 |
NA |
NA |
NA |
NA |
TTD |
| GLB1 |
1-Naphthalenesulfonic acid, 3-hydroxy-4-(2-(1-hydroxy-2-naphthalenyl)diazenyl)- |
NA |
600000 |
NA |
NA |
NA |
NA |
TTD |
| GLB1 |
2-[(3,5-Diiodo-4-oxidophenyl)(3,5-diiodo-4-oxocyclohexa-2,5-dien-1-ylidene)methyl]benzoate |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| GLB1 |
(1S,7R)-1,7,8,9,10,10-hexachloro-4-(2,4-dinitroanilino)-4-azatricyclo[5.2.1.02,6]dec-8-ene-3,5-dione |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GLB1 |
5-Methylene-piperidine-3,4-diol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GLB1 |
1-Butyl-5-methyl-piperidine-3,4-diol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GLB1 |
5-Methoxy-piperidine-3,4-diol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GLB1 |
2-(2,2-Dihydroxy-ethyl)-pyrrolidine-3,4-diol |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| GLB1 |
[(1S,2R,6S,8S)-10,10-dimethyl-3,7,9,11-tetraoxa-4-azatricyclo[6.3.0.02,6]undec-4-en-5-yl]methanol |
NA |
150000|1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| GLB1 |
5-[(2S,3S,4R)-3,4-dihydroxypyrrolidin-2-yl]-N-isopropyl-2-methyl-3-furamide |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GLB1 |
4-[2-(2,4-Difluoro-phenylamino)-thiazol-4-yl]-benzene-1,2-diol |
NA |
320000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |