| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GHSR |
(2S)-2-[(2S)-2-(2-aminoacetamido)-3-hydroxypropanamido]-2-{[(1S)-1-carbamoyl-2-phenylethyl]carbamoyl}ethyl heptanoate |
NA |
889000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GHSR |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| GHSR |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| GHSR |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
| GHSR |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| GHSR |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| GK |
Adenylyl Imidodiphosphate |
900000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| GK |
[[(2R,3S,4R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy-hydroxyphosphoryl]oxy-(arsonomethyl)phosphinic acid |
2900000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| GK |
Adenosine Triphosphate |
200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| GK |
Adenosine-5'-(Beta, Gamma-Methylene)Triphosphate |
300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| GLA |
5-Methylpiperidine-3,4-diol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GLA |
D-Galacto-Isofagomine |
2000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GLA |
(2R,3S,4S,5S)-2-Hydroxymethyl-piperidine-3,4,5-triol |
NA |
920000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GLA |
(2R,3S,4S,5R)-2-Hydroxymethyl-piperidine-3,4,5-triol |
NA |
390000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GLA |
(2R,3R,4S,5S)-2-(aminomethyl)-5-(hydroxymethyl)pyrrolidine-3,4-diol |
NA |
266000 |
NA |
NA |
NA |
NA |
BindingDB |
| GLA |
(3R,4S,5R,6R)-6-(4-aminobutyl)-5-(hydroxymethyl)piperidine-3,4-diol |
2000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GLA |
(3R,4S,5R,6R)-6-(2-hydroxyethyl)-5-(hydroxymethyl)piperidine-3,4-diol |
2000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GLA |
N-[4-[(2R,3R,4S,5R)-4,5-dihydroxy-3-(hydroxymethyl)piperidin-2-yl]butyl]-5-(dimethylamino)naphthalene-1-sulfonamide |
2000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GLA |
(2R,3S,4R)-2-[[4-[4-(hydroxymethyl)phenyl]triazol-1-yl]methyl]pyrrolidine-3,4-diol |
NA |
159000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GLA |
(2R,3S,4R)-2-[[4-(4-methoxyphenyl)triazol-1-yl]methyl]pyrrolidine-3,4-diol |
NA |
185000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |