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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
GGPS1 [1-Hydroxy-3-(pyridin-3-yl)propane-1,1-diyl]bis(phosphonic acid) NA 410000 NA NA NA NA BindingDB
GGPS1 Minodronic Acid NA 107150 NA NA NA NA BindingDB|PubChem
GGPS1 Bisphosphonate, 60 NA 169820 NA NA NA NA BindingDB
GGPS1 Bisphosphonate, 56 NA 107150 NA NA NA NA BindingDB
GGPS1 Phosphonic acid, (1-hydroxybutylidene)di- NA 620000 NA NA NA NA BindingDB
GGPS1 Alendronic Acid NA 436520|440000|398107 NA NA NA NA BindingDB|PubChem
GGPS1 Bph-715 NA 250000 NA NA NA NA BindingDB
GGPS1 Bisphosphonate, 58 NA 117490 NA NA NA NA BindingDB
GGPS1 Bisphosphonate, 59 NA 141250 NA NA NA NA BindingDB
GGPS1 Bisphosphonate, 63 NA 316230 NA NA NA NA BindingDB
GGPS1 [2-(4-Aminophenyl)-1-hydroxy-1-phosphonoethyl]phosphonic acid NA 180000 NA NA NA NA BindingDB
GGPS1 (1-Hydroxy-2-phenyl-1-phosphonoethyl)phosphonic acid NA 220000 NA NA NA NA BindingDB
GGPS1 4-(2-Hydroxy-2,2-bis-phosphono-ethylsulfanyl)-pyridinium NA 550000 NA NA NA NA BindingDB
GGPS1 1-Hydroxypentane-1,1-bisphosphonate NA 200000 NA NA NA NA BindingDB
GGPS1 2-[Methyl-(4-methyl-pent-3-enyl)-amino]-ethyl-diphosphate NA 240000 NA NA NA NA BindingDB
GGPS1 Pamidronic Acid NA 180000|181970|199526 NA NA NA NA BindingDB|PubChem
GGPS1 [1-Hydroxy-2-(1H-imidazol-4-yl)-1-phosphono-ethyl]-phosphonic acid NA 220000 NA NA NA NA BindingDB
GGPS1 Risedronic Acid NA|8300000 331130|350000|300000000|NA NA NA NA NA BindingDB|PubChem
GGPS1 NE97220 NA 220000 NA NA NA NA BindingDB
GGPS1 2-[(Bis-phosphono-methyl)-amino]-4-methyl-pyridinium NA 260000 NA NA NA NA BindingDB