| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GBA1 |
(3R,4R,5R)-1-[(4-fluorophenyl)methyl]-5-(hydroxymethyl)piperidine-3,4-diol |
111800 |
269800 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
(1R,2S,3S,4R,5S,6R)-5,6-di(nonoxy)cyclohexane-1,2,3,4-tetrol |
NA |
144000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
(2R,3S,4R,5S,6S)-5-[2-[(2S,3S,4R,5S,6R)-4,5-dihydroxy-2-(hydroxymethyl)-6-methoxyoxan-3-yl]sulfanylpyridin-3-yl]oxy-6-(hydroxymethyl)-2-methoxyoxane-3,4-diol |
5500000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
N-Methyl-1-Deoxynojirimycin |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
(2R,3R,4R,5S)-2-(hydroxymethyl)-1-propylpiperidine-3,4,5-triol |
NA |
700000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA2 |
L-Ido-1-Deoxynojirimycin |
NA |
400000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA2 |
Miglustat |
NA |
180000 |
NA |
NA |
NA |
NA |
PubChem |
| GBA2 |
(2S,3S)-1-[5-(1-adamantylmethoxy)pentyl]-2-(hydroxymethyl)piperidin-3-ol |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA2 |
(2R,3R,4S)-1-butyl-2-(hydroxymethyl)piperidine-3,4-diol |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA2 |
(2R,3S)-1-butyl-2-(hydroxymethyl)-3,6-dihydro-2H-pyridin-3-ol |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA2 |
(2R,3R)-1-[5-(1-adamantylmethoxy)pentyl]-2-(hydroxymethyl)-3,6-dihydro-2H-pyridin-3-ol |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA3 |
N-(2,3,4-Trihydroxy-5-hydroxymethyl-cyclohexyl)-acetamide |
NA |
14000000000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA3 |
1-Deoxynojirimycin |
NA |
240000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| GBA3 |
(2S,3S,4S,5R)-2-Hydroxymethyl-piperidine-3,4,5-triol |
NA |
980000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA3 |
2,5-Dideoxy-2,5-Imino-D-Glucitol |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA3 |
Validamine |
NA |
130000000000 |
NA |
NA |
NA |
NA |
BindingDB |
| GCGR |
3-[2-(1H-Benzoimidazol-2-ylsulfanyl)-acetyl]-benzoic acid |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GCGR |
2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3-hydroxy-phenyl)-ethanone |
380000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GCGR |
1-(3,4-Dihydroxy-phenyl)-2-(1-methyl-1H-benzoimidazol-2-ylsulfanyl)-ethanone |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GCGR |
4-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3,4-dihydroxy-phenyl)-butan-1-one |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |