| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GCGR |
5-[2-(1H-Benzoimidazol-2-ylsulfanyl)-acetyl]-2-hydroxy-benzoic acid |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GCGR |
1-(3,4-Dihydroxy-phenyl)-2-(4,5-diphenyl-1H-imidazol-2-ylsulfanyl)-ethanone |
180000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GCGR |
1-(3,4-Dihydroxy-phenyl)-2-(1H-imidazol-2-ylsulfanyl)-ethanone |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GCGR |
4-[2-(1H-Benzoimidazol-2-ylsulfanyl)-acetyl]-benzoic acid |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GCGR |
1-(3,4-Dihydroxy-phenyl)-2-(quinolin-2-ylsulfanyl)-ethanone |
160000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GCGR |
4-[2-(1H-benzoimidazol-2-ylsulfanyl)-1-hydroxy-ethyl]-2-chloro-phenol |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GCGR |
2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3,4-dihydroxy-phenyl)-pentan-1-one |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GCGR |
1-[4-[1-[3-(3,5-Dichlorophenyl)-5-(6-methoxynaphthalen-2-yl)pyrazol-1-yl]ethyl]benzoyl]pyrrolidine-3-carboxylic acid |
NA |
131100 |
NA |
NA |
NA |
NA |
TTD |
| GCGR |
2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3-chloro-4-hydroxy-phenyl)-ethanone O-methyl-oxime |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GCGR |
2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3-chloro-4-hydroxy-phenyl)-ethanone O-benzyl-oxime |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GCGR |
2-(1H-Benzimidazol-2-ylsulfanyl)-1-phenylethanone |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GCGR |
2-(1,3-Benzoxazol-2-ylsulfanyl)-1-(3,4-dihydroxyphenyl)ethanone |
250000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GCGR |
2-(1H-benzimidazol-2-ylsulfanyl)-1-(3,5-dihydroxyphenyl)ethanone |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GCGR |
2-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-(3,4-dichlorophenyl)ethan-1-one |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GCGR |
2-(1H-benzimidazol-2-ylsulfanyl)-1-(3,4-dimethoxyphenyl)ethanone |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GDA |
3-Benzyl-3H-imidazo[4,5-e][1,4]diazepine-6,8-dione |
227000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GFPT1 |
Aaptamine |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| GGCT |
Ggstop |
170000 |
NA |
NA |
NA |
NA |
NA |
GtoPDB |
| GGH |
(2S)-2-{[hydroxy(methyl)phosphoryl]amino}pentanedioic acid |
930000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| GGH |
(2S)-2-{[hydroxy(phenyl)phosphoryl]amino}pentanedioic acid |
950000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |