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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
GGPS1 Bisphpshonate-943 NA 120000 NA NA NA NA BindingDB
GGPS1 Bisphpshonate-942 NA 440000 NA NA NA NA BindingDB
GGPS1 Neridronic Acid NA 690000 NA NA NA NA BindingDB|PubChem
GGPS1 (3-Amino-1-hydroxy-1-phosphono-butyl)-phosphonic acid NA 330000 NA NA NA NA BindingDB
GGT1 (S)-2-Amino-5-boronopentanoic acid 3820000 NA NA NA NA NA BindingDB
GGT1 (2R)-2-(2-aminoethylamino)-4-boronobutanoic acid 260000 NA NA NA NA NA BindingDB
GGT1 (2R)-4-borono-2-[[4-(phenylsulfamoyl)phenyl]methylamino]butanoic acid 173000 NA NA NA NA NA BindingDB
GGT1 (2R)-2-[[(2R)-2-aminopropyl]amino]-4-boronobutanoic acid 254000 NA NA NA NA NA BindingDB
GGT1 (2R)-4-borono-2-[(4-methoxyphenyl)methylamino]butanoic acid 343000 NA NA NA NA NA BindingDB
GGT1 (2R)-4-borono-2-(2-phenylethylamino)butanoic acid 220000|356000 NA NA NA NA NA BindingDB
GGT1 3-[[[(1R)-3-borono-1-carboxypropyl]amino]methyl]benzoic acid 589000 NA NA NA NA NA BindingDB
GGT1 (2R)-4-borono-2-(3-phenylpropylamino)butanoic acid 108000 NA NA NA NA NA BindingDB
GGT1 (2R)-2-[[(2R)-2-amino-3-phenylpropyl]amino]-4-boronobutanoic acid 508000 NA NA NA NA NA BindingDB
GGT1 (2R)-2-(benzylamino)-4-boronobutanoic acid 202000|2150000 NA NA NA NA NA BindingDB
GGT1 2-Amino-4-borono-2-ethylbutanoic acid 444000|874000 NA NA NA NA NA BindingDB
GGT1 2-Amino-2-(2-boronoethyl)pentanoic acid 198000|703000 NA NA NA NA NA BindingDB
GGT1 N-(5-(4-methoxybenzyl)-1,3,4-thiadiazol-2-yl)benzenesulfonamide 376000 NA NA NA NA NA BindingDB
GHSR Imipenem NA NA NA NA NA 300000 PubChem
GHSR Cefazolin NA NA NA NA NA 300000 PubChem
GHSR Meropenem NA NA NA NA NA 300000 PubChem