| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRM1 |
(S)-2-amino-5-phosphonopentanoic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
D-2-aminoadipic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM1 |
alpha-Amino-3-(hydroxy)-5-methyl-4-isoxazoleacetic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM1 |
(2R,1''S,2''R)-2-(2''-sulfonocyclopropyl)glycine |
254000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R,1''R,2''S)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R,1''R,2''R)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2S,1''S,2''S)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R,1''S,2''S)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2S,1''R,2''R)-2-(2''-sulfonocyclopropyl)glycine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2S)-2-amino-4-phosphonobutanoic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
Aida |
NA|214000 |
214000|NA |
NA |
NA |
NA |
NA |
PubChem |
| GRM1 |
(A+-)-1-Amino-cis-cyclopentane-1,3-dicarboxylic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM1 |
D-Glutamic Acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
PubChem|TTD |
| GRM1 |
2-Amino-3-(4-bromo-3-hydroxyisoxazol-5-YL)propanoic acid |
329000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2S,3S)-3-(carboxymethyl)azetidine-2-carboxylic acid |
NA |
NA |
NA |
210000 |
NA |
NA |
TTD |
| GRM1 |
Glutamic Acid |
NA |
NA |
NA |
156000 |
NA |
NA |
PubChem |
| GRM1 |
2-Amino-2-(4-phosphonophenyl)propanoic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
homo-AMPA |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM1 |
(2R,4R)-4-Amino-1-(3-chloro-benzyl)-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM1 |
(2R,4R)-4-Amino-1-biphenyl-2-ylmethyl-pyrrolidine-2,4-dicarboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |