| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GRM5 |
2-Amino-4-(4-hydroxy-[1,2,5]thiadiazol-3-yl)-butyric acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM6 |
2-Aminoheptanedioic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM6 |
Kainic acid |
NA |
NA |
NA |
299000 |
NA |
NA |
BindingDB|TTD |
| GRM6 |
(2R,4R)-1,4-Diamino-pyrrolidine-2,4-dicarboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM6 |
(1R,2S,4R,5S)-2-Amino-bicyclo[2.1.1]hexane-2,5-dicarboxylic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM6 |
(1S,2S,4S,5R)-2-Amino-bicyclo[2.1.1]hexane-2,5-dicarboxylic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM6 |
2-Amino-6-(3-hydroxy-5-methyl-isoxazol-4-yl)-hexanoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM6 |
(1R,2S,4R,5R)-2-Amino-bicyclo[2.1.1]hexane-2,5-dicarboxylic acid |
NA |
NA |
NA |
800000 |
NA |
NA |
BindingDB|TTD |
| GRM6 |
2-Amino-2,3-methano-4-phosphonobutanoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM6 |
(S)-Ampa |
NA |
NA |
NA |
220000 |
NA |
NA |
BindingDB|TTD |
| GRM6 |
D-2-aminoadipic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM6 |
(1R,2S)-1-amino-2-(phosphonomethyl)cyclopropanecarboxylic acid |
NA |
NA |
NA |
111000 |
NA |
NA |
BindingDB|TTD |
| GRM6 |
alpha-Amino-3-(hydroxy)-5-methyl-4-isoxazoleacetic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| GRM6 |
D-Glutamic Acid |
NA |
NA |
NA |
270000|1000000 |
NA |
NA |
BindingDB|PubChem|TTD |
| GRM6 |
(2S,3S)-3-(carboxymethyl)azetidine-2-carboxylic acid |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GRM6 |
Glutamic Acid |
NA |
NA |
NA |
270000 |
NA |
NA |
PubChem |
| GRM6 |
2-Amino-2-(4-phosphonophenyl)propanoic acid |
480000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRM6 |
Quisqualic Acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GRM6 |
(2S)-2-amino-3-(3,5-dioxo-1,2,4-oxadiazolidin-4-yl)-2-methylpropanoic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GRM6 |
2-Amino-bicyclo[3.2.0]heptane-2,7-dicarboxylic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |