| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GUCY1B1 |
Gemfibrozil |
NA |
NA |
NA |
624000 |
NA |
NA |
PubChem |
| GUSB |
2-Phenyl-4(3H)-Quinazolinone |
NA |
177000 |
NA |
NA |
NA |
NA |
TTD |
| GUSB |
2-(4-Methylphenyl)quinazolin-4(3H)-one |
NA |
172700 |
NA |
NA |
NA |
NA |
TTD |
| GUSB |
2-(3,4,5-Trimethoxyphenyl)quinazolin-4-ol |
NA |
120500 |
NA |
NA |
NA |
NA |
TTD |
| GUSB |
2-(3-hydroxyphenyl)quinazolin-4(3H)-one |
NA |
198200 |
NA |
NA |
NA |
NA |
TTD |
| GUSB |
N,N-bis(3,5-dimethylpyrazol-1-ylmethyl)-cyclohexylamine |
NA |
456600 |
NA |
NA |
NA |
NA |
TTD |
| GYPA |
(2R,3S,5R,6S)-5-(benzyloxy)-6-(benzyloxymethyl)-2-(hydroxymethyl)tetrahydro-2H-pyran-3-ol |
NA |
NA |
2400000 |
NA |
NA |
NA |
BindingDB |
| GYPA |
(1S,3R,5S,6R,8S,11R,13S,15R,16S,18R)-6-(hydroxymethyl)-11-methyl-15-phenylmethoxy-16-(phenylmethoxymethyl)-2,7,12,17-tetraoxatetracyclo[9.8.0.03,8.013,18]nonadecan-5-ol |
NA |
NA |
240000 |
NA |
NA |
NA |
BindingDB |
| GYPA |
Desulfated yessotoxin |
NA |
NA |
270000 |
NA |
NA |
NA |
BindingDB |
| GYPA |
[(1R,3S,5R,7S,9R,11S,13R,14S,16R,18S,20R,22S,25R,27S,30S,31R,33S,35R,37S,40S,42R,44S,46R,48S)-40-[(2R,3E)-2-hydroxy-5-methylideneocta-3,7-dien-2-yl]-13,25,27,30,35-pentamethyl-39-methylidene-13-(2-sulfonatooxyethyl)-4,8,12,17,21,26,32,36,41,45,49-undecaoxaundecacyclo[25.22.0.03,25.05,22.07,20.09,18.011,16.031,48.033,46.035,44.037,42]nonatetracontan-14-yl] sulfate |
NA |
NA |
120000 |
NA |
NA |
NA |
BindingDB |
| HAGH |
S-(N-Methyl-N-hydroxycarbomyl)ethylglutathione |
426000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| HAO1 |
Ethyl 5-((2-chlorophenyl)thio)-1H-1,2,3-triazole-4-carboxylate |
NA |
251000 |
NA |
NA |
NA |
NA |
BindingDB |
| HAO1 |
Ethyl 5-((2-fluorophenyl)thio)-1H-1,2,3-triazole-4-carboxylate |
NA |
430000 |
NA |
NA |
NA |
NA |
BindingDB |
| HAO1 |
5-phenyl-1H-1,2,3-triazole-4-carboxylic acid |
NA |
4079500 |
NA |
NA |
NA |
NA |
BindingDB |
| HAVCR2 |
2-methyl-5H,6H-(1,2,4)triazolo(1,5-c)quinazolin-5-one |
NA |
NA |
810000 |
NA |
NA |
NA |
ChEMBL |
| HAVCR2 |
2-(propan-2-yl)-5H,6H-[1,2,4]triazolo[1,5-c]quinazolin-5-one |
NA |
NA |
330000 |
NA |
NA |
NA |
ChEMBL |
| HAVCR2 |
9-methoxy-2-propan-2-yl-6H-[1,2,4]triazolo[1,5-c]quinazolin-5-one |
NA |
NA |
250000 |
NA |
NA |
NA |
ChEMBL |
| HAVCR2 |
4-Amino-8-chloroquinoline-3-carboxylic acid |
NA |
NA |
130000 |
NA |
NA |
NA |
ChEMBL |
| HAVCR2 |
2-Benzimidazolinethione, 5-chloro- |
NA |
NA |
670000 |
NA |
NA |
NA |
ChEMBL |
| HAVCR2 |
(4-Methylphenyl)(1-methylpyrazolo[4,5-e]pyrimidin-4-yl)amine |
NA |
NA |
850000 |
NA |
NA |
NA |
ChEMBL |