| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| HAVCR2 |
4-([1,2,4]Triazolo[3,4-b][1,3,4]thiadiazol-6-yl)aniline |
NA |
NA |
740000 |
NA |
NA |
NA |
ChEMBL |
| HAVCR2 |
2-Methyl-4-oxazolo[4,5-b]pyridin-2-yl-phenylamine |
NA |
NA |
460000 |
NA |
NA |
NA |
ChEMBL |
| HAVCR2 |
2-Mercapto-4,6-dimethylnicotinonitrile |
NA |
NA |
780000 |
NA |
NA |
NA |
ChEMBL |
| HAVCR2 |
2-Methyl-1,5,6,7-tetrahydrocyclopenta[d]pyrimidine-4-thione |
NA |
NA |
450000 |
NA |
NA |
NA |
ChEMBL |
| HAVCR2 |
1,3-Dimethyl-6-m-tolylamino-1H-pyrimidine-2,4-dione |
NA |
NA |
1400000 |
NA |
NA |
NA |
ChEMBL |
| HAVCR2 |
3-[2-(dimethylamino)ethyl]-2-thioxo-2,3-dihydroquinazolin-4(1H)-one |
NA |
NA |
530000 |
NA |
NA |
NA |
ChEMBL |
| HCAR1 |
3-Bromo-5-hydroxybenzoic acid |
NA |
NA |
NA |
129000 |
NA |
NA |
BindingDB|TTD |
| HCAR1 |
3-Cyano-5-hydroxybenzoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HCAR1 |
3-t-Butyl-5-hydroxybenzoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HCAR1 |
3-Carboxy-5-hydroxypyridine 1-oxide |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HCAR1 |
(3-hydroxyphenyl)boronic Acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HCAR1 |
3-hydroxy-5-(trifluoromethyl)benzoic Acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HCAR1 |
5-Hydroxynicotinic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HCAR1 |
5-Hydroxy-3-phenylbenzoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HCAR1 |
3,5-Dihydroxyphenylphosphonic Acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HCAR1 |
3,5-Dihydroxyphenyl(Methyl)Phosphinic Acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HCAR1 |
5-(2H-tetrazol-5-yl)benzene-1,3-diol |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HCAR1 |
3-Hydroxybenzoic acid |
NA |
NA |
NA |
184000 |
NA |
NA |
BindingDB|TTD |
| HCAR1 |
3,5-Dihydroxybenzoic Acid |
NA |
NA |
NA |
377000|191000 |
NA |
NA |
BindingDB|GtoPDB|TTD |
| HCAR1 |
3-Hydroxy-5-methoxybenzoic acid |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |