| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| HCK |
2-Aminoquinoline |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HCK |
1-[2-(Furan-2-yl)pyrrolidin-1-yl]prop-2-en-1-one |
1250000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HCN1 |
2-methoxy-N-{[1-(morpholin-4-yl)cyclohexyl]methyl}benzamide |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| HCN1 |
2-methoxy-N-[2-(4-methylpiperazin-1-yl)ethyl]benzamide |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| HCN1 |
2-chloro-N-[[1-(4-methylpiperazin-1-yl)cyclohexyl]methyl]benzamide |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| HCN1 |
2-ethoxy-N-[[1-(4-phenylpiperazin-1-yl)cyclohexyl]methyl]benzamide |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| HCN1 |
2-hydroxy-N-[[2-(4-methylpiperazin-1-yl)-1,3-dihydroinden-2-yl]methyl]benzamide |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| HCN1 |
2-ethyl-N-[[1-(4-propan-2-ylpiperazin-1-yl)cyclohexyl]methyl]benzamide |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| HCN4 |
Mel57A |
NA |
NA |
NA |
103780 |
NA |
NA |
BindingDB|TTD |
| HCN4 |
3-[(Z)-4-[[(Z)-4-(7,8-dimethoxy-2-oxo-1H-3-benzazepin-3-yl)but-2-enyl]-[(2S)-2-(3,4-dimethoxyphenyl)propyl]amino]but-2-enyl]-7,8-dimethoxy-1H-3-benzazepin-2-one |
NA |
NA |
NA |
135730 |
NA |
NA |
BindingDB|TTD |
| HCN4 |
2-methoxy-N-[(2-piperidin-1-yl-1,3-dihydroinden-2-yl)methyl]benzamide |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| HCN4 |
N-[[2-(4-methylpiperazin-1-yl)-1,3-dihydroinden-2-yl]methyl]-2-(trifluoromethoxy)benzamide |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| HCN4 |
2-fluoro-N-[[2-(4-methylpiperazin-1-yl)-1,3-dihydroinden-2-yl]methyl]benzamide |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| HCN4 |
2-methyl-N-[[1-(4-methylpiperazin-1-yl)cyclohexyl]methyl]benzamide |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| HCN4 |
3-methoxy-N-[[2-(4-methylpiperazin-1-yl)-1,3-dihydroinden-2-yl]methyl]benzamide |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| HCN4 |
2-chloro-N-[[2-(4-methylpiperazin-1-yl)-1,3-dihydroinden-2-yl]methyl]benzamide |
NA |
158489.32 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| HCN4 |
2-hydroxy-N-[[2-(4-methylpiperazin-1-yl)-1,3-dihydroinden-2-yl]methyl]benzamide |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| HCN4 |
4-methoxy-N-[[2-(4-methylpiperazin-1-yl)-1,3-dihydroinden-2-yl]methyl]benzamide |
NA |
199526.23 |
NA |
NA |
NA |
NA |
TTD |
| HCRTR1 |
N-cyclopropyl-2-(2,5-dimethyl-1H-indol-3-yl)-N-(pyridin-3-ylmethyl)acetamide |
1000000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| HCRTR1 |
G-N-H-A-A-G-I-L-T-L |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |