| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| HCRTR2 |
R-S-G-P-P-G-L-Q-G-R |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HCRTR2 |
SB-334867 |
NA |
835000 |
NA |
NA |
NA |
NA |
BindingDB |
| HCRTR2 |
H-Pyr-Pro-Leu-Pro-Asp-Cys-Cys-Arg-Gln-Lys-Thr-Cys-Ser-OH |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HCRTR2 |
H-Pyr-Pro-Leu-Pro-Asp-Cys-Cys-Arg-Gln-Lys-Thr-OH |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HDAC1 |
N-acetyl-S-(N-benzylthiocarbamoyl)-l-cysteine |
NA |
3440000 |
NA |
NA |
NA |
NA |
BindingDB |
| HDAC1 |
Butanoate |
NA|365000 |
140000|800000|NA |
NA |
NA |
NA |
NA |
BindingDB |
| HDAC1 |
7-Methanesulfonyl-heptanoic acid phenylamide |
NA |
230000 |
NA |
NA |
NA |
NA |
BindingDB |
| HDAC1 |
6-(hydrazinecarbonylamino)-N-phenylhexanamide |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| HDAC1 |
6-Methanesulfonylamino-hexanoic acid phenylamide |
NA |
7500000 |
NA |
NA |
NA |
NA |
BindingDB |
| HDAC1 |
Acetylcysteine |
NA |
3160000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| HDAC1 |
4-Methylquinoline-8-thiol |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| HDAC1 |
5-Methylquinoline-8-thiol |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| HDAC1 |
(1E,6E)-1,7-bis[4-[(2E)-3,7-dimethylocta-2,6-dienoxy]-3-methoxyphenyl]-4-[(2E)-3,7-dimethylocta-2,6-dienyl]hepta-1,6-diene-3,5-dione |
NA |
217000 |
NA |
NA |
NA |
NA |
BindingDB |
| HDAC1 |
(1E,6E)-1,7-bis[4-[(2E)-3,7-dimethylocta-2,6-dienoxy]-3-methoxyphenyl]-4,4-bis[(2E)-3,7-dimethylocta-2,6-dienyl]hepta-1,6-diene-3,5-dione |
NA |
786000 |
NA |
NA |
NA |
NA |
BindingDB |
| HDAC1 |
(1E,6E)-1,7-bis[3-methoxy-4-[(2E,6E)-3,7,11-trimethyldodeca-2,6,10-trienoxy]phenyl]hepta-1,6-diene-3,5-dione |
NA |
122000 |
NA |
NA |
NA |
NA |
BindingDB |
| HDAC1 |
(1E,6E)-1-[4-[(2E)-3,7-dimethylocta-2,6-dienoxy]-3-methoxyphenyl]-7-(4-hydroxy-3-methoxyphenyl)hepta-1,6-diene-3,5-dione |
NA |
495000 |
NA |
NA |
NA |
NA |
BindingDB |
| HDAC1 |
(1E,6E)-1,7-bis[4-[(2E)-3,7-dimethylocta-2,6-dienoxy]-3-methoxyphenyl]hepta-1,6-diene-3,5-dione |
NA |
188000 |
NA |
NA |
NA |
NA |
BindingDB |
| HDAC1 |
(2R)-2-acetamido-3-[3-[[(2R)-2-acetamido-2-carboxyethyl]sulfanylcarbothioylamino]propylcarbamothioylsulfanyl]propanoic acid |
NA |
5960000 |
NA |
NA |
NA |
NA |
BindingDB |
| HDAC1 |
(2R)-2-acetamido-3-[4-[[(2R)-2-acetamido-2-carboxyethyl]sulfanylcarbothioylamino]butylcarbamothioylsulfanyl]propanoic acid |
NA |
2330000 |
NA |
NA |
NA |
NA |
BindingDB |
| HDAC1 |
(2R)-2-acetamido-3-[[5-[[(2R)-2-acetamido-2-carboxyethyl]sulfanylcarbothioylamino]-4-methylpentyl]carbamothioylsulfanyl]propanoic acid |
NA |
2190000 |
NA |
NA |
NA |
NA |
BindingDB |