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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
HDAC1 Tanespimycin NA 1000000 NA NA NA NA PubChem
HDAC1 Tubacin NA NA NA 217000 NA NA BindingDB
HDAC1 Caffeic Acid NA 2540000 NA NA NA NA BindingDB|PubChem
HDAC1 3-[[(E)-3-[4-(dimethylamino)phenyl]prop-2-enoyl]amino]-N-hydroxypropanamide NA 250000 NA NA NA NA TTD
HDAC1 2-Azidoethyl 8-[4-[(3-azido-5-methoxyphenyl)methoxy]anilino]-8-oxooctanoate NA 111000 NA NA NA NA BindingDB|TTD
HDAC1 Ubenimex NA 1000000 NA NA NA NA PubChem
HDAC1 (E)-N-(2-amino-4-methylphenyl)-3-[3-methoxy-4-[2-(4-methoxyanilino)-2-oxoethoxy]phenyl]prop-2-enamide NA 118000 NA NA NA NA BindingDB
HDAC1 (2R)-2-[(1-hydroxy-6-sulfanylidenepyridine-2-carbonyl)amino]propanoic acid NA 270000 NA NA NA NA BindingDB|TTD
HDAC1 Valproic acid hydroxamate NA 560000 NA NA NA NA BindingDB|TTD
HDAC1 (E)-N-(2-amino-4-methylphenyl)-3-[4-methoxy-3-[2-(4-methoxyanilino)-2-oxoethoxy]phenyl]prop-2-enamide NA 164610 NA NA NA NA BindingDB
HDAC1 (E)-N-(2-amino-4-methylphenyl)-3-[3-[2-[3-bromo-5-(trifluoromethyl)anilino]-2-oxoethoxy]-4-methoxyphenyl]prop-2-enamide NA 124670 NA NA NA NA BindingDB
HDAC1 Bml-210 NA 120000 NA NA NA NA BindingDB
HDAC1 Hexanediamide, N-(2-aminophenyl)-N'-phenyl- NA 238000 NA NA NA NA BindingDB
HDAC1 Heptanediamide, N,N'-diphenyl- NA 204000 NA NA NA NA BindingDB
HDAC1 N'-(3-aminophenyl)-N-phenylheptanediamide NA 500000 NA NA NA NA BindingDB
HDAC1 N'-(4-aminophenyl)-N-phenyloctanediamide NA 186000 NA NA NA NA BindingDB
HDAC1 N'-(4-aminophenyl)-N-phenylheptanediamide NA 123000 NA NA NA NA BindingDB
HDAC1 N-phenyl-N'-pyridin-2-ylheptanediamide NA 140000 NA NA NA NA BindingDB
HDAC1 N'-(2-methoxyphenyl)-N-phenyloctanediamide NA 470000 NA NA NA NA BindingDB
HDAC1 N'-(4-methoxyphenyl)-N-phenylheptanediamide NA 438000 NA NA NA NA BindingDB