Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| HDAC1 | N'-(2,4-dimethoxyphenyl)-N-phenylheptanediamide | NA | 387000 | NA | NA | NA | NA | BindingDB |
| HDAC1 | 8-Mercaptoquinoline | NA | 200000 | NA | NA | NA | NA | TTD |
| HDAC1 | Curcumin | NA | 115000|187000 | NA | NA | NA | NA | BindingDB|PubChem |
| HDAC1 | N-Acetyl-S-[N-(2-phenylethyl)thiocarbamoyl]-L-cysteine | NA | 3450000 | NA | NA | NA | NA | BindingDB |
| HDAC1 | N-(2-Amino-5-fluorophenyl)-4-[[[1-oxo-3-(3-pyridinyl)-2-propen-1-yl]amino]methyl]benzamide | NA | 260000 | NA | NA | NA | NA | BindingDB|PubChem |
| HDAC10 | Acetylcysteine | NA | 3160000 | NA | NA | NA | NA | PubChem |
| HDAC10 | Chlorogenic Acid | NA | 375000|200000 | NA | NA | NA | NA | PubChem |
| HDAC10 | Butyric Acid | 136000 | NA | NA | NA | NA | NA | PubChem |
| HDAC10 | Valproic Acid | 564000|NA | NA|995000|7240000 | NA | NA | NA | NA | PubChem |
| HDAC10 | Sodium Butyrate | NA|365000 | 140000|NA|800000 | NA | NA | NA | NA | PubChem |
| HDAC10 | (1E,4Z,6E)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-one | NA | 115000 | NA | NA | NA | NA | PubChem |
| HDAC10 | Tanespimycin | NA | 1000000 | NA | NA | NA | NA | PubChem |
| HDAC10 | Caffeic Acid | NA | 2540000 | NA | NA | NA | NA | PubChem |
| HDAC10 | Curcumin | NA | 187000 | NA | NA | NA | NA | PubChem |
| HDAC11 | 6-[[4-(benzenesulfonyl)-5-oxido-1,2,5-oxadiazol-5-ium-3-yl]oxy]-N-hydroxyhexanamide | NA | 608000 | NA | NA | NA | NA | BindingDB |
| HDAC11 | Acetylcysteine | NA | 3160000 | NA | NA | NA | NA | PubChem |
| HDAC11 | 4-[[2,4-dioxo-3-(2-phenylethyl)quinazolin-1-yl]methyl]-N-hydroxythiophene-2-carboxamide | NA | 128900 | NA | NA | NA | NA | BindingDB |
| HDAC11 | Chlorogenic Acid | NA | 375000|200000 | NA | NA | NA | NA | PubChem |
| HDAC11 | Butyric Acid | 136000 | NA | NA | NA | NA | NA | PubChem |
| HDAC11 | Valproic Acid | NA|564000 | 995000|NA|7240000 | NA | NA | NA | NA | PubChem |