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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
HDAC4 N-(5-phenyl-1,3-thiazol-2-yl)-7-[(3,3,3-trifluoro-2,2-dihydroxypropanoyl)amino]heptanamide NA 2500000 NA NA NA NA BindingDB
HDAC4 N-(4-bromophenyl)-7-[(3,3,3-trifluoro-2,2-dihydroxypropanoyl)amino]heptanamide NA 2600000 NA NA NA NA BindingDB
HDAC4 N-(4-methoxyphenyl)-7-[(3,3,3-trifluoro-2,2-dihydroxypropanoyl)amino]heptanamide NA 1600000 NA NA NA NA BindingDB
HDAC4 N-(1,3-benzothiazol-2-yl)-7-[(3,3,3-trifluoro-2,2-dihydroxypropanoyl)amino]heptanamide NA 430000 NA NA NA NA BindingDB
HDAC4 N-[5-(4-bromophenyl)-1,3-thiazol-2-yl]-7-[(3,3,3-trifluoro-2,2-dihydroxypropanoyl)amino]heptanamide NA 1700000 NA NA NA NA BindingDB
HDAC4 N-[5-(4-hydroxyphenyl)-1,3-thiazol-2-yl]-7-[(3,3,3-trifluoro-2,2-dihydroxypropanoyl)amino]heptanamide NA 2300000 NA NA NA NA BindingDB
HDAC4 N-(5-methoxy-1,3-benzothiazol-2-yl)-7-[(3,3,3-trifluoro-2,2-dihydroxypropanoyl)amino]heptanamide NA 1900000 NA NA NA NA BindingDB
HDAC4 N-(4-phenylphenyl)-7-[(3,3,3-trifluoro-2,2-dihydroxypropanoyl)amino]heptanamide NA 1100000 NA NA NA NA BindingDB
HDAC4 Chlorogenic Acid NA 375000|200000 NA NA NA NA PubChem
HDAC4 NA 125000 NA NA NA NA BindingDB
HDAC4 Butyric Acid 136000|NA NA|2000000 NA NA NA NA PubChem|TTD
HDAC4 N-hydroxy-4-phenylbutanamide NA 140000 NA NA NA NA BindingDB|TTD
HDAC4 Valproic Acid NA|564000 1000000|995000|7240000|2000000|NA NA NA NA NA BindingDB|PubChem|TTD
HDAC4 N-hydroxybutanamide NA 2000000 NA NA NA NA TTD
HDAC4 Entinostat NA 142000 NA NA NA NA BindingDB|PubChem
HDAC4 N-(2-aminophenyl)-7,7-di(1H-indol-3-yl)heptanamide NA 150000 NA NA NA NA BindingDB|TTD
HDAC4 Phenylbutyric acid NA 2000000 NA NA NA NA PubChem|TTD
HDAC4 Sodium Butyrate NA|365000 140000|NA|800000 NA NA NA NA PubChem
HDAC4 (1E,4Z,6E)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-one NA 115000 NA NA NA NA PubChem
HDAC4 Vorinostat NA 12000000 NA NA NA NA BindingDB|PubChem