| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| HDAC4 |
RG-2833 |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| HDAC4 |
Tanespimycin |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| HDAC4 |
Caffeic Acid |
NA |
2540000 |
NA |
NA |
NA |
NA |
PubChem |
| HDAC4 |
(3S,6Z,9S,12R,16S)-6-ethylidene-16-[(E)-4-methylsulfanylbut-1-enyl]-9-(methylsulfanylmethyl)-3,12-di(propan-2-yl)-1-oxa-4,7,10-triazacyclohexadecane-2,5,8,11,14-pentone |
NA |
110000 |
NA |
NA |
NA |
NA |
TTD |
| HDAC4 |
(1S,2S)-N-hydroxy-2-phenylcyclopropane-1-carboxamide |
NA |
904000 |
NA |
NA |
NA |
NA |
TTD |
| HDAC4 |
Valproic acid hydroxamate |
NA |
170000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| HDAC4 |
(1S,5S,6R,9S,15E,20R)-20-butyl-5-hydroxy-6-(2-methylpropyl)-2-oxa-11,12-dithia-7,19,22-triazabicyclo[7.7.6]docos-15-ene-3,8,18,21-tetrone |
NA |
132500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| HDAC4 |
N1-(2-Aminophenyl)-N7-phenylheptanediamide |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |
| HDAC4 |
Curcumin |
NA |
187000 |
NA |
NA |
NA |
NA |
PubChem |
| HDAC5 |
Acetylcysteine |
NA |
3160000 |
NA |
NA |
NA |
NA |
PubChem |
| HDAC5 |
HDAC6/Tubulin Inhibitor MPT0B451 |
NA |
356000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| HDAC5 |
N-[3-[4-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methylcarbamoyl]-5-methylpyrazol-1-yl]phenyl]-N'-hydroxyoctanediamide |
NA |
101000 |
NA |
NA |
NA |
NA |
BindingDB |
| HDAC5 |
Chlorogenic Acid |
NA |
375000|200000 |
NA |
NA |
NA |
NA |
PubChem |
| HDAC5 |
Butyric Acid |
136000|NA |
NA|2000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| HDAC5 |
Valproic Acid |
NA|564000 |
1000000|995000|7240000|NA|2000000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| HDAC5 |
N-hydroxybutanamide |
NA |
360000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| HDAC5 |
Phenylbutyric acid |
NA |
2000000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| HDAC5 |
Sodium Butyrate |
NA|365000 |
140000|NA|800000 |
NA |
NA |
NA |
NA |
PubChem |
| HDAC5 |
(1E,4Z,6E)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-one |
NA |
115000 |
NA |
NA |
NA |
NA |
PubChem |
| HDAC5 |
RG-2833 |
NA |
180000 |
NA |
NA |
NA |
NA |
TTD |