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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
HSPA8 Ethyl 1-[2-(2-chloro-6-fluorophenyl)acetyl]piperidine-4-carboxylate NA 999000 NA NA NA NA BindingDB
HSPA8 N-(4-chlorophenyl)-N'-(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)urea NA 999000 NA NA NA NA BindingDB
HSPA8 3-(2,5-dimethyl-1H-pyrrol-1-yl)benzoic acid NA 999000 NA NA NA NA BindingDB
HSPA8 N-[2,3-bis(furan-2-yl)quinoxalin-6-yl]azepane-1-carboxamide NA 999000 NA NA NA NA BindingDB
HSPA8 N-(5-methyl-1,2-oxazol-3-yl)-2-quinazolin-4-ylsulfanylacetamide NA 999000 NA NA NA NA BindingDB
HSPA8 8-(2-methylpropoxycarbonyl)-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-4-carboxylic acid NA 164000 NA NA NA NA BindingDB
HSPA8 8-(2-ethoxycarbonylphenoxy)carbonyl-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-4-carboxylic acid NA 112000 NA NA NA NA BindingDB
HSPA8 8-((2-(Methoxycarbonyl)phenoxy)carbonyl)-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-4-carboxylic acid NA 115000 NA NA NA NA BindingDB
HSPA8 N-(4-methoxybenzo[d]thiazol-2-yl)-5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-amine NA 999000 NA NA NA NA BindingDB
HSPA8 5-[(5-Bromo-2-methoxyphenyl)methylidene]-2-(furan-2-yl)-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one NA 999000 NA NA NA NA BindingDB
HSPA8 3-(2-furyl)-N-(3-methoxypropyl)-3-{[(4-methylphenyl)sulfonyl]amino}propanamide NA 999000 NA NA NA NA BindingDB
HSPA8 6-methyl-8-nitro-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-4-carboxylic acid NA 117000 NA NA NA NA BindingDB
HSPA8 3-Amino-N-phenylphthalimide NA 999000 NA NA NA NA BindingDB
HSPA8 8-chloro-6-hydroxy-9-nitro-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-4-carboxylic acid NA 175000 NA NA NA NA BindingDB
HSPA8 2-(4-cyano-3-propylpyrido[1,2-a]benzimidazol-1-yl)sulfanyl-N-(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)acetamide NA 999000 NA NA NA NA BindingDB
HSPA8 5'-Deoxyadenosine NA NA 130000|131826 NA NA NA BindingDB
HSPA8 [4-[(2-Hydroxybenzoyl)diazenyl]anilino] benzoate NA 999000 NA NA NA NA BindingDB
HSPA8 2-Methyl-4-(4-methylquinolin-8-yl)-4-azatricyclo[5.2.1.02,6]dec-8-ene-3,5-dione NA 999000 NA NA NA NA BindingDB
HSPA8 NA 999000 NA NA NA NA BindingDB
HSPA8 4-[2-(2-chloro-5-nitrophenyl)vinyl]-6-(trifluoromethyl)-2(1H)-pyrimidinone NA 999000 NA NA NA NA BindingDB