| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| HSPE1 |
Pentamidine |
NA |
250000 |
NA |
NA |
NA |
NA |
PubChem |
| HSPE1 |
Nifurtimox |
NA |
250000 |
NA |
NA |
NA |
NA |
PubChem |
| HTR1A |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR1A |
8-(4-Benzylpiperazin-1-yl)-4-phenyl-5-thia-1,7-diazatricyclo[7.3.0.02,6]dodeca-2(6),3,7,9,11-pentaene |
NA |
389045.14 |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
(4-Fluorophenyl)-[4-(3-thia-1,7-diazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaen-8-yl)piperazin-1-yl]methanone |
NA |
102329.3 |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
8-[4-[(4-Chlorophenyl)-phenylmethyl]piperazin-1-yl]-3-thia-1,7-diazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaene |
NA |
204173.79 |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
8-(4-Benzylpiperazin-1-yl)-4,5-dimethyl-3-thia-1,7-diazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaene |
NA |
125892.54 |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
1-[2-hydroxy-3-methyl-4-[[4-[4-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone |
3020000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
5,6-Methylenedioxy-N,N-diisopropyltryptamine |
NA |
933000 |
NA |
NA |
NA |
NA |
BindingDB |
| HTR1A |
4-(4,5-dihydro-1H-imidazol-2-ylmethyl)-3-fluorobenzene-1,2-diol;hydrochloride |
NA |
64565422903466 |
NA |
NA |
NA |
NA |
BindingDB |
| HTR1A |
(1R)-3-[3-(3,4-difluorophenyl)-6,7-dihydro-4H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-1-phenylpropan-1-ol |
330400 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
3-[3-(4-Benzylpiperazin-1-yl)-2-hydroxypropyl]-5-(4-fluorophenyl)-5-methylimidazolidine-2,4-dione |
377500 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
3-[3-(4-Benzhydrylpiperazin-1-yl)-2-hydroxypropyl]-5-methyl-5-naphthalen-1-ylimidazolidine-2,4-dione |
413200 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
4-[hydroxy(1H-imidazol-2-yl)methyl]benzene-1,2-diol;hydrochloride |
NA |
2290867652768 |
NA |
NA |
NA |
NA |
BindingDB |
| HTR1A |
4-(1H-imidazol-2-ylmethyl)benzene-1,2-diol;hydrochloride |
NA |
162181|346737|660693|812831|1548817 |
NA |
NA |
NA |
NA |
BindingDB |
| HTR1A |
4-(4,5-dihydro-1H-imidazol-2-ylmethyl)-5-fluorobenzene-1,2-diol;hydrochloride |
NA |
36307805477010 |
NA |
NA |
NA |
NA |
BindingDB |
| HTR1A |
5-(4,5-dihydro-1H-imidazol-2-ylmethyl)-3-fluorobenzene-1,2-diol;hydrochloride |
NA |
54954087385763 |
NA |
NA |
NA |
NA |
BindingDB |
| HTR1A |
4-[(2-Chlorophenyl)sulfonylmethyl]-6-(4-methylpiperazin-1-yl)-1,3,5-triazin-2-amine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1A |
methyl (2S)-2-[(2S,3R,5S,12bR)-3-ethenyl-5-oxido-1,2,3,4,6,7,12,12b-octahydroindolo[2,3-a]quinolizin-5-ium-2-yl]-3-hydroxypropanoate |
NA |
NA |
NA |
500000 |
NA |
NA |
TTD |
| HTR1A |
N-[[5-bromo-2-[(4-methylphenyl)methoxy]phenyl]methyl]-1-phenylethanamine |
195600 |
NA |
NA |
NA |
NA |
NA |
TTD |