Navigator

      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
HTR1A 4-Methylthiodimethyltryptamine NA 151000 NA NA NA NA BindingDB
HTR1A 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(3''-chlorophenyl)piperazine 1130000 NA NA NA NA NA TTD
HTR1A 5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(3''-chlorophenyl)piperazine 5000000 NA NA NA NA NA TTD
HTR1A 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(3''-trifluoromethylphenyl)piperazine 2874000 NA NA NA NA NA TTD
HTR1A 2{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(2''-methoxyphenyl)piperazine 1241000 NA NA NA NA NA TTD
HTR1A 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(2''-methoxyphenyl)piperazine 756000 NA NA NA NA NA TTD
HTR1A 5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(2''-methoxyphenyl)piperazine 5000000 NA NA NA NA NA TTD
HTR1A 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(4''-fluorophenyl)piperazine 800000 NA NA NA NA NA TTD
HTR1A 5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(4''-fluorophenyl)piperazine 5000000 NA NA NA NA NA TTD
HTR1A 2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(2''-pyrimidil)piperazine 656000 NA NA NA NA NA TTD
HTR1A 4-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(2''-pyrimidyl)piperazine 558000 NA NA NA NA NA TTD
HTR1A 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-4-(3''-methyl)piperazine 5000000 NA NA NA NA NA TTD
HTR1A 5-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}pentyl-4-(N-methyl)piperazine 5000000 NA NA NA NA NA TTD
HTR1A 3-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}propyl-(3,4-dihydroisoquinoline) 1124000 NA NA NA NA NA TTD
HTR1A 4{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-(3,4-dihydroisoquinoline) 1331000 NA NA NA NA NA TTD
HTR1A 2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-(6,7-dimethoxy-3,4-dihydroisoquinoline) 5000000 NA NA NA NA NA TTD
HTR1A 4-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-(6,7-dimethoxy-3,4-dihydroisoquinoline) 5000000 NA NA NA NA NA TTD
HTR1A 2-{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}ethyl-4-(3''-chlorophenyl)piperazine 686000 NA NA NA NA NA TTD
HTR1A 4{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(3''-trifluoromethylphenyl)piperazine 5000000 NA NA NA NA NA TTD
HTR1A 4{2-[2-(3-Methoxyphenyl)ethyl]phenoxy}butyl-4-(4''-fluorophenyl)piperazine 5000000 NA NA NA NA NA TTD