| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| HTR1A |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
| HTR1A |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| HTR1A |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR1B |
1-[2-hydroxy-3-methyl-4-[[4-[4-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone |
3580000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1B |
3-[(dipropylamino)methyl]-5-methoxy-N,N-dipropyl-2,4-dihydrochromen-3-amine |
NA |
138038|138038.43 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| HTR1B |
Benzyl-{1-[2-fluoro-3-(5-[1,2,4]triazol-4-yl-1H-indol-3-yl)-propyl]-piperidin-4-yl}-methyl-amine |
NA |
NA |
NA |
103000 |
NA |
NA |
BindingDB|TTD |
| HTR1D |
1-[2-hydroxy-3-methyl-4-[[4-[4-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone |
2400000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1E |
1-[2-hydroxy-3-methyl-4-[[4-[4-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone |
5370000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR1E |
2-(4-fluorophenyl)-3-(4-methoxyphenyl)-5,6,7,7a-tetrahydro-3H-pyrrolo[1,2-c]imidazol-1-one |
NA |
441000000 |
NA |
NA |
NA |
NA |
BindingDB |
| HTR1F |
1-[2-hydroxy-3-methyl-4-[[4-[4-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone |
2970000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR2A |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR2A |
1-[2-hydroxy-3-methyl-4-[[4-[4-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone |
7470000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR2A |
DL-methamphetamine |
101000 |
NA |
NA |
NA |
NA |
NA |
PubChem|TTD |
| HTR2A |
2-methyl-5,6,7,8-tetrahydro-4H-[1,2]oxazolo[4,5-d]azepin-3-one |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR2A |
2-ethyl-5,6,7,8-tetrahydro-4H-[1,2]oxazolo[4,5-d]azepin-3-one |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR2A |
3-methoxy-5,6,7,8-tetrahydro-4H-[1,2]oxazolo[4,5-d]azepine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR2A |
2,6-Dimethyl-4,5,7,8-tetrahydro-[1,2]oxazolo[4,5-d]azepin-3-one |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR2A |
2-Ethyl-6-methyl-4,5,7,8-tetrahydro-[1,2]oxazolo[4,5-d]azepin-3-one |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR2A |
2,4-Pyrimidinediamine, 5-[5-iodo-4-methoxy-2-(1-methylethyl)phenoxy]- |
100000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR2A |
5,6,7,8-tetrahydro-4H-isoxazolo(4,5-d)azepin-3-ol |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |