| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| HTR2A |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR2A |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR2A |
3-[(dipropylamino)methyl]-5-methoxy-N,N-dipropyl-2,4-dihydrochromen-3-amine |
NA |
213796.21 |
NA |
NA |
NA |
NA |
TTD |
| HTR2A |
Pramoxine |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR2A |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR2A |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR2A |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
| HTR2A |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| HTR2A |
2-Ethyl-4,5,6,7-tetrahydro-[1,2]oxazolo[5,4-c]pyridin-3-one |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HTR2A |
3-Ethoxy-4,5,6,7-tetrahydro-[1,2]oxazolo[5,4-c]pyridine |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HTR2A |
3-Methoxy-6-methyl-4,5,7,8-tetrahydro-[1,2]oxazolo[4,5-d]azepine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR2A |
3-Ethoxy-6-methyl-4,5,7,8-tetrahydro-[1,2]oxazolo[4,5-d]azepine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR2A |
2-Methyl-4,5,6,7-tetrahydro-[1,2]oxazolo[4,5-c]pyridin-3-one |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HTR2A |
2-Ethyl-4,5,6,7-tetrahydro-[1,2]oxazolo[4,5-c]pyridin-3-one |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HTR2A |
2-Benzyl-4,5,6,7-tetrahydro-[1,2]oxazolo[4,5-c]pyridin-3-one |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HTR2A |
2-benzyl-5,6,7,8-tetrahydro-4H-[1,2]oxazolo[4,5-c]azepin-3-one |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HTR2A |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR2B |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR2B |
1-[2-hydroxy-3-methyl-4-[[4-[4-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone |
3300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR2B |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |