| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| HTR2C |
2,6-Dimethyl-4,5,7,8-tetrahydro-[1,2]oxazolo[4,5-d]azepin-3-one |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR2C |
2-Ethyl-6-methyl-4,5,7,8-tetrahydro-[1,2]oxazolo[4,5-d]azepin-3-one |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR2C |
5,6,7,8-tetrahydro-4H-isoxazolo(4,5-d)azepin-3-ol |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR2C |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR2C |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR2C |
5-Methoxy-1',4'-dipropylspiro[2,4-dihydrochromene-3,2'-piperazine] |
NA |
468000 |
NA |
NA |
NA |
NA |
BindingDB |
| HTR2C |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR2C |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR2C |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
| HTR2C |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| HTR2C |
Thymol |
NA |
NA |
NA |
NA |
NA |
170000 |
PubChem |
| HTR2C |
2-Ethyl-4,5,6,7-tetrahydro-[1,2]oxazolo[5,4-c]pyridin-3-one |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HTR2C |
3-Ethoxy-4,5,6,7-tetrahydro-[1,2]oxazolo[5,4-c]pyridine |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HTR2C |
3-Methoxy-6-methyl-4,5,7,8-tetrahydro-[1,2]oxazolo[4,5-d]azepine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR2C |
3-Ethoxy-6-methyl-4,5,7,8-tetrahydro-[1,2]oxazolo[4,5-d]azepine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR2C |
2-Methyl-4,5,6,7-tetrahydro-[1,2]oxazolo[4,5-c]pyridin-3-one |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HTR2C |
2-Ethyl-4,5,6,7-tetrahydro-[1,2]oxazolo[4,5-c]pyridin-3-one |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HTR2C |
2-Benzyl-4,5,6,7-tetrahydro-[1,2]oxazolo[4,5-c]pyridin-3-one |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HTR2C |
2-benzyl-5,6,7,8-tetrahydro-4H-[1,2]oxazolo[4,5-c]azepin-3-one |
NA |
NA |
NA |
1000000 |
NA |
NA |
TTD |
| HTR2C |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |