| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| HTR2C |
2-{methyl[2-(morpholin-4-yl)-2-oxoethyl]amino}-1-(2-phenyl-1H-indol-3-yl)ethan-1-one |
NA |
213796|214000|213796.21 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| HTR3A |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR3A |
2,4-Pyrimidinediamine, 5-[5-iodo-4-methoxy-2-(1-methylethyl)phenoxy]- |
100000000 |
NA |
NA |
NA |
NA|NA |
NA|NA |
BindingDB|TTD |
| HTR3A |
Eucalyptol |
NA |
257040|257039.58 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| HTR3A |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR3A |
cis-1-Methyl-5-(phenylethynyl)-3-(piperidin-1-ylmethyl)pyrrolidin-2-one |
NA |
251188.64 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| HTR3A |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR3A |
(1R,3R,8S,10R,13S,16S,17R)-8-tert-butyl-6,12,17-trihydroxy-16-methyl-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,18-trione |
NA |
730000|3900000 |
NA |
NA |
NA |
NA |
GtoPDB |
| HTR3A |
(4aS,5R,10bR)-5-phenyl-1,2,3,4,4a,5,6,10b-octahydrobenzo[h]isoquinoline-7,8-diol |
870000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| HTR3A |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR3A |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR3A |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |
| HTR3A |
Carumonam |
NA |
NA |
NA |
NA |
NA |
500000 |
PubChem |
| HTR3A |
Linalool, (+/-)- |
NA |
141254|141253.75 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| HTR3A |
Doripenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HTR3A |
Bilobalide |
NA |
470000|3100000 |
NA |
NA |
NA |
NA |
GtoPDB |
| HTR3B |
(1R,3R,8S,10R,13S,16S,17R)-8-tert-butyl-6,12,17-trihydroxy-16-methyl-2,4,14,19-tetraoxahexacyclo[8.7.2.01,11.03,7.07,11.013,17]nonadecane-5,15,18-trione |
NA |
3900000 |
NA |
NA |
NA |
NA |
GtoPDB |
| HTR3B |
Bilobalide |
NA |
3100000 |
NA |
NA |
NA |
NA |
GtoPDB |
| HTR4 |
1-[2-hydroxy-3-methyl-4-[[4-[4-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone |
6310000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR5A |
1-[2-hydroxy-3-methyl-4-[[4-[4-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone |
6900000 |
NA |
NA |
NA |
NA |
NA |
TTD |