| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| HTR6 |
1-[2-hydroxy-3-methyl-4-[[4-[4-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone |
1790000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR6 |
2,4-Pyrimidinediamine, 5-[5-iodo-4-methoxy-2-(1-methylethyl)phenoxy]- |
100000000 |
NA |
NA |
NA |
NA|NA |
NA|NA |
BindingDB|TTD |
| HTR6 |
N-[4-(3,4-dihydro-1H-isoquinolin-2-yl)butyl]quinoline-8-sulfonamide |
41858718 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| HTR6 |
6-chloro-3-(1-propylpiperidin-4-yl)-1H-benzimidazol-2-one |
NA |
580000 |
NA |
NA |
NA |
NA |
TTD |
| HTR7 |
Ikonnikoside I |
NA |
135000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| HTR7 |
1-[2-hydroxy-3-methyl-4-[[4-[4-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone |
3980000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR7 |
1-Acetoxy-9,17-octadecadiene-12,14-diyne-11,16-diol |
NA |
118100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| HTR7 |
Dihydrobaicalin |
NA |
179000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| HTR7 |
2-[6-[4-(4-Methoxyphenyl)piperazin-1-yl]hexyl]benzo[de]isoquinoline-1,3-dione |
116500 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| HTR7 |
2-[[4-[[4-(4-Chlorophenyl)piperazin-1-yl]methyl]phenyl]methyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one |
201400 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| HTR7 |
(E)-3-(butylthio)-N-((6,7-dimethoxy-3,4-dihydroisoquinolin-2(1H)-yl)methylene)-1H-inden-5-amine |
300000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| HTR7 |
(S)-8-hydroxy-1-methoxy-, Z-9-heptadecene-4,6-diyn-3-one |
NA |
150000 |
NA |
NA |
NA |
NA |
TTD |
| HTR7 |
(4aS,5R,10bR)-5-phenyl-1,2,3,4,4a,5,6,10b-octahydrobenzo[h]isoquinoline-7,8-diol |
220000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| HTR7 |
Falcarindiol |
NA |
117500 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| HTR7 |
Baicalein |
NA |
350000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| HTR7 |
Wogonin |
NA |
350000 |
NA |
NA |
NA |
NA |
TTD |
| HTR7 |
N-[4-(6,7-dihydro-4H-thieno[3,2-c]pyridin-5-yl)butyl]quinoline-3-sulfonamide |
506829 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| HTR7 |
(Z)-Butylidenephthalide |
NA |
126600 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| HTR7 |
Baicalin |
NA |
200000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| HTT |
(2S)-1-[(2S)-6-amino-2-[butyl(hydroxy)phosphoryl]oxyhexanoyl]pyrrolidine-2-carboxylic acid |
NA |
23300000 |
NA |
NA |
NA |
NA |
BindingDB |