| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| IARS1 |
(S)-1-[2-(3-Hydroxy-4-methoxy-benzoylamino)-ethoxycarbonyl]-2-methyl-butyl-ammonium |
NA |
106000 |
NA |
NA |
NA |
NA |
BindingDB |
| IARS1 |
(1S,2S)-1-[(2R,3S,4R,5R)-5-(6-Amino-purin-9-yl)-3,4-dihydroxy-tetrahydro-furan-2-ylmethoxycarbonyl]-2-methyl-butyl-ammonium |
NA |
183000 |
NA |
NA |
NA |
NA |
BindingDB |
| IARS1 |
(2S,3S)-2-amino-N-[[(2R,3S,4R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl-hydroxysulfamoyl]-3-methylpentanamide |
NA |
132000 |
NA |
NA |
NA |
NA |
BindingDB |
| ICAM1 |
Indole |
NA |
NA |
300000 |
NA |
NA |
NA |
PubChem |
| ICMT |
(2R)-3-[(2E)-3,7-dimethylocta-2,6-dienyl]sulfanyl-2-[(2-phenoxybenzoyl)amino]propanoic acid |
NA |
149000 |
NA |
NA |
NA |
NA |
BindingDB |
| ICMT |
(2R)-2-[(2-phenoxybenzoyl)amino]-3-undecylsulfanylpropanoic acid |
NA |
210000 |
NA |
NA |
NA |
NA |
BindingDB |
| IDH1 |
3-[(3-methoxy-4-pyrrol-1-ylanilino)methyl]-6,7-dimethyl-1H-quinolin-2-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| IDH1 |
N-cyclohexyl-2-(N-(3-fluorophenyl)-2-(2-methyl-1H-imidazol-1-yl)acetamido)-2-(o-tolyl)acetamide |
NA |
NA |
608000 |
NA |
NA |
NA |
BindingDB |
| IDH1 |
Mutant IDH1 inhibitor |
NA |
NA |
140000|142000 |
NA |
NA |
NA |
BindingDB |
| IDO1 |
6-Fluoro-3-((1E)-2-(3-pyridinyl)ethenyl)-1H-indole |
NA |
350000|477600 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
Naphthalene-1,2,4-trione |
NA |
675000 |
NA |
NA |
NA |
NA |
BindingDB |
| IDO1 |
9-Fluorenone |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| IDO1 |
1-[2-(2,4-Dichlorophenyl)-2-methoxyethyl]imidazole |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
(3-Aminonaphthalen-2-yl)methanol |
NA |
190000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
4-Hydroxycarbazole |
NA |
400000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
3-(1H-Imidazol-4-yl)benzaldehyde |
NA |
825000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
4-(1H-Imidazol-5-yl)pyridine |
NA |
1800000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
4-(2-Thienyl)-1H-imidazole |
NA |
422000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
Tryptamine |
160000|156000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| IDO1 |
4-(1H-indol-3-ylmethyl)-1,3-thiazole |
1292000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |